SCHEMBL7417006

SCHEMBL7417006

c1cc(-c2ncc[nH]2)cc(-n2cnc3cc(-c4ccoc4)cnc32)c1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NT5E P21589 2/20 0.45
GAK O14976 2/20 0.39
CDK8 P49336 1/20 0.36
KDR P35968 1/20 0.35
MTOR P42345 1/20 0.35
ADK P55263 1/20 0.35
NISCH Q9Y2I1 1/20 0.35
HPGD P15428 1/20 0.32
PRKCI P41743 3/20 0.32
CCNT1 O60563 1/20 0.31
CCNA2 P20248 1/20 0.31
CDK2 P24941 1/20 0.31
CDK9 P50750 1/20 0.31
CSF1R P07333 1/20 0.31
FYN P06241 3/20 0.31
PIM1 P11309 1/20 0.30
MRGPRX4 Q96LA9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6799283 0.82 NT5E (0.47) NT5EGAKKDRFYN
SCHEMBL6804619 0.79 NT5E (0.69) NT5EGAKCDK8KDRHPGD
SCHEMBL6797821 0.78 NT5E (0.47) NT5EGAKKDR
SCHEMBL6803619 0.76 GABRG2 (0.52) NT5EGAKCDK8KDR
SCHEMBL6804409 0.76 NT5E (0.44) NT5EGAKCDK8KDRHPGD
SCHEMBL6796978 0.75 NT5E (0.45) NT5EGAKCDK8KDRHPGD
SCHEMBL6803865 0.74 NT5E (0.42) NT5EGAKCDK8KDRHPGD
SCHEMBL6799281 0.73 NT5E (0.43) NT5EGAKKDRHPGD
SCHEMBL6798778 0.73 NT5E (0.45) NT5EGAKKDRHPGD
SCHEMBL6807826 0.72 NT5E (0.44) NT5EGAKCDK8KDRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214319-A1 IMIDAZO-PYRIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS Merck Sharp & Dohme Limited (GB) 2002-06-19 EP disclosed
WO-2001018000-A1 IMIDAZO-PYRIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 2001-03-15 WO disclosed