SCHEMBL6803097

SCHEMBL6803097

C[Si](C)(C)O[C@@H]1C[C@@H](CO)N(C(=O)OCc2ccccc2)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.43
HTR2C P28335 1/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PSEN1 P49768 1/20 0.41
PSEN2 P49810 1/20 0.41
APH1B Q8WW43 1/20 0.41
NCSTN Q92542 1/20 0.41
APH1A Q96BI3 1/20 0.41
PSENEN Q9NZ42 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PDK1 Q15118 1/20 0.41
PDK2 Q15119 1/20 0.41
PDK3 Q15120 1/20 0.41
PDK4 Q16654 1/20 0.41
PREP P48147 1/20 0.41
NPC1L1 Q9UHC9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18962 0.89 ABCB1 (0.43) POLBHTR2CMEN1KMT2ANPSR1
SCHEMBL8833139 0.89 ABCB1 (0.43) POLBHTR2CMEN1KMT2ANPSR1
SCHEMBL29254 0.89 ABCB1 (0.43) POLBHTR2CMEN1KMT2ANPSR1
SCHEMBL15958482 0.89 ABCB1 (0.43) POLBHTR2CMEN1KMT2ANPSR1
SCHEMBL9026282 0.89 ABCB1 (0.43) POLBHTR2CMEN1KMT2ANPSR1
SCHEMBL6796832 0.89 PREP (0.43) POLBHTR2CMEN1KMT2ANPSR1
SCHEMBL6319947 0.87 POLB (0.45) POLBHTR2CNPSR1PSEN1PSEN2
SCHEMBL30645964 0.85 ABCB1 (0.42) POLBHTR2CPSEN1PSEN2APH1B
SCHEMBL30054860 0.85 ABCB1 (0.44) POLBHTR2CPSEN1PSEN2APH1B
SCHEMBL18569430 0.85 ABCB1 (0.44) POLBHTR2CPSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6833456-B2 Heterocyclic sulfides such as 5-(2-(2R-Hydroxymethyl-pyrrolidine-1-carbonyl)-thieno(3,2-b)pyridin-7 -ylamino)-2-methyl-indole-1-carboxylic acid methylamide, used as angiogenesis inhibitors AGOURON PHARMACEUTICALS, INC. 2004-12-21 US disclosed