SCHEMBL6804774

SCHEMBL6804774

O=C1c2ccccc2CCN1OCc1ccc(C(F)(F)F)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.46
HTR2A P28223 2/20 0.46
HTR2C P28335 2/20 0.46
HTR2B P41595 2/20 0.46
SIGMAR1 Q99720 2/20 0.46
SCN1A P35498 1/20 0.46
SCN5A Q14524 1/20 0.46
SCN9A Q15858 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.44
KDM4E B2RXH2 1/20 0.44
HTT P42858 1/20 0.44
MEN1 O00255 1/20 0.43
POLB P06746 1/20 0.43
GAA P10253 1/20 0.43
KMT2A Q03164 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
CHRM5 P08912 1/20 0.42
DRD1 P21728 1/20 0.41
DRD3 P35462 1/20 0.41
CA12 O43570 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24055077 0.83 KMT2A (0.45) DRD2MEN1POLBGAAKMT2A
SCHEMBL29500334 0.78 DRD2 (0.54) DRD2HTR2AHTR2CHTR2BSIGMAR1
SCHEMBL15846180 0.76 KMT2A (0.65) HTTMEN1POLBGAAKMT2A
SCHEMBL15467684 0.74 NR1H2 (0.42) HTR2AHTR2CHTR2BSIGMAR1KMT2A
SCHEMBL16914914 0.71 IDO1 (0.47) SCN1ASCN5ASCN9AKDM4EKMT2A
SCHEMBL30199163 0.71 KMT2A (0.49) HTR2AMEN1POLBGAAKMT2A
SCHEMBL2025017 0.69 KMT2A (0.55) DRD2HTR2AHTR2CHTR2BSIGMAR1
SCHEMBL28922536 0.69 KMT2A (0.64) DRD2MEN1POLBGAAKMT2A
SCHEMBL30232651 0.69 KMT2A (0.64) DRD2MEN1POLBGAAKMT2A
SCHEMBL28865189 0.69 KMT2A (0.47) SMN1; SMN2KDM4EMEN1POLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6818774-B2 2-(S)-(6-(4-FLUORO-BENZYLOXY)-3-OXO-3,4-DIHYDRO-1H-ISOQUINOLIN -2-YL)- PROPIONAMIDE FOR EXAMPLE; ALZHEIMER'S DISEASE OR SENILE DEMENTIA HOFFMAN-LA ROCHE INC. 2004-11-16 US disclosed