SCHEMBL6805728

SCHEMBL6805728

NC(=O)c1cccc2nc(-c3ccc(N4CCNCC4)nc3)[nH]c12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.53
AURKB Q96GD4 2/20 0.53
KDR P35968 1/20 0.52
PARP1 P09874 6/20 0.45
KCNH2 Q12809 3/20 0.43
DGAT1 O75907 1/20 0.43
IKBKE Q14164 1/20 0.42
TBK1 Q9UHD2 1/20 0.42
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
CACNA1C Q13936 1/20 0.41
ASIC3 Q9UHC3 1/20 0.41
JAK2 O60674 1/20 0.41
PRKCA P17252 1/20 0.41
PRKCQ Q04759 1/20 0.41
PRKCD Q05655 1/20 0.41
PDE10A Q9Y233 1/20 0.40
ATR Q13535 1/20 0.40
GPR119 Q8TDV5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6812407 0.96 AURKA (0.50) AURKAAURKBKDRPARP1KCNH2
SCHEMBL6805914 0.92 AURKA (0.55) AURKAAURKBKDRPARP1KCNH2
SCHEMBL6806391 0.91 AURKA (0.54) AURKAAURKBKDRPARP1KCNH2
SCHEMBL6809975 0.91 AURKA (0.54) AURKAAURKBKDRPARP1KCNH2
SCHEMBL6806351 0.89 AURKA (0.59) AURKAAURKBKDRPARP1KCNH2
SCHEMBL6802984 0.89 JAK2 (0.53) AURKAAURKBKDRPARP1KCNH2
SCHEMBL6805042 0.88 AURKA (0.57) AURKAAURKBKDRPARP1KCNH2
SCHEMBL6810290 0.86 AURKA (0.54) AURKAAURKBKDRPARP1KCNH2
SCHEMBL6805101 0.86 AURKA (0.64) AURKAAURKBKDRPARP1KCNH2
SCHEMBL6810130 0.85 AURKA (0.54) AURKAAURKBKDRPARP1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696437-B1 Heterocyclically substituted benzimidazoles, the production and application thereof ABBOTT GMBH & CO. KG (DE) 2004-02-24 US disclosed