SCHEMBL6806962

SCHEMBL6806962

NC(=O)c1cccc2[nH]c(-c3cccnc3)nc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKN1 Q16512 3/20 1.00
PKN2 Q16513 3/20 1.00
PARP1 P09874 17/20 0.88
PARP2 Q9UGN5 2/20 0.88
DHODH Q02127 2/20 0.88
PLK4 O00444 1/20 0.74
MAPK13 O15264 1/20 0.74
DYRK3 O43781 1/20 0.74
ROCK2 O75116 1/20 0.74
RPS6KA5 O75582 1/20 0.74
PRKD3 O94806 1/20 0.74
MAP4K4 O95819 1/20 0.74
CHEK2 O96017 1/20 0.74
PIM1 P11309 1/20 0.74
PHKG2 P15735 1/20 0.74
PRKACA P17612 1/20 0.74
RPS6KB1 P23443 1/20 0.74
CSNK1D P48730 1/20 0.74
CLK2 P49760 1/20 0.74
GSK3A P49840 1/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29411982 1.00 PKN1 (1.00) PKN1PKN2PARP1PARP2DHODH
SCHEMBL656979 0.88 PKN1 (0.78) PKN1PKN2PARP1PARP2DHODH
SCHEMBL7561483 0.88 PKN1 (0.79) PKN1PKN2PARP1PARP2DHODH
SCHEMBL657818 0.85 PKN1 (0.73) PKN1PKN2PARP1PARP2DHODH
SCHEMBL6809991 0.85 PKN1 (1.00) PKN1PKN2PARP1PARP2DHODH
SCHEMBL458836 0.85 PARP1 (1.00) PKN1PKN2PARP1PARP2DHODH
SCHEMBL29412034 0.85 PARP1 (1.00) PKN1PKN2PARP1PARP2DHODH
SCHEMBL6809904 0.84 PKN1 (0.74) PKN1PKN2PARP1PARP2DHODH
SCHEMBL505358 0.82 PARP1 (1.00) PKN1PKN2PARP1PARP2DHODH
SCHEMBL6586688 0.81 PKN1 (0.68) PKN1PKN2PARP1PARP2DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101353342-A 2-pyridinyl-1H-benzimidazole-4-acidamide type derivative UNIV SHANGHAI JIAOTONG (CN) 2009-01-28 CN disclosed
US-6696437-B1 Heterocyclically substituted benzimidazoles, the production and application thereof ABBOTT GMBH & CO. KG (DE) 2004-02-24 US disclosed