SCHEMBL681189

SCHEMBL681189

C=C(C(C)C)[C@H](CNC(C)C)c1cc(F)cc(F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 8/20 0.40
ADRB1 P08588 7/20 0.40
ADRB3 P13945 6/20 0.40
TSHR P16473 3/20 0.37
HIF1A Q16665 2/20 0.37
ADRA1A P35348 2/20 0.37
MEN1 O00255 2/20 0.36
LMNA P02545 2/20 0.36
KMT2A Q03164 2/20 0.36
BLM P54132 2/20 0.36
APEX1 P27695 1/20 0.36
MAPT P10636 3/20 0.34
MTOR P42345 2/20 0.34
KDM4E B2RXH2 2/20 0.34
MAPK1 P28482 2/20 0.34
HSD17B10 Q99714 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL681754 0.90 ADRB2 (0.35) ADRB2ADRB1ADRB3TSHRHIF1A
SCHEMBL680060 0.84 ADRB2 (0.44) ADRB2ADRB1ADRB3TSHRHIF1A
SCHEMBL681274 0.84 ADRB2 (0.40) ADRB2ADRB1ADRB3TSHRHIF1A
SCHEMBL684339 0.82 ADRB2 (0.41) ADRB2ADRB1ADRB3TSHRHIF1A
SCHEMBL680064 0.80 PDPK1 (0.44) ADRB2ADRB1ADRB3TSHRHIF1A
SCHEMBL681163 0.80 TACR1 (0.37) ADRB2ADRB1ADRB3TSHRHIF1A
SCHEMBL17803796 0.78 ADRB2 (0.41) ADRB2ADRB1ADRB3TSHRHIF1A
SCHEMBL17803797 0.78 ADRB2 (0.38) ADRB2ADRB1ADRB3TSHRHIF1A
SCHEMBL681539 0.77 AKT1 (0.44) ADRB2ADRB1ADRB3TSHRHIF1A
SCHEMBL680197 0.77 ADRB2 (0.40) ADRB2ADRB1ADRB3TSHRHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9359340-B2 Hydroxylated and methoxylated pyrimidyl cyclopentanes as Akt protein kinase inhibitors ARRAY BIOPHARMA INC. (US) 2016-06-07 US disclosed
US-8063050-B2 Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors ARRAY BIOPHARMA INC. (US) 2011-11-22 US disclosed