SCHEMBL681259

SCHEMBL681259

C=C(C(C)C)[C@H](CNC(C)(C)C)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 3/20 0.40
CNR2 P34972 2/20 0.38
LDHA P00338 2/20 0.38
LDHB P07195 2/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
TSHR P16473 1/20 0.36
NFKB1 P19838 1/20 0.36
HIF1A Q16665 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL681467 0.86 CNR2 (0.41) ADRB2CNR2LDHALDHBLMNA
SCHEMBL681594 0.84 CA1 (0.38) CNR2LDHALDHBCA1CA2
SCHEMBL681564 0.84 CA1 (0.38) CNR2LDHALDHBCA1CA2
SCHEMBL17803813 0.84 HPGD (0.40) ADRB2CYP1A2CYP2D6TSHRNFKB1
SCHEMBL684762 0.82 CNR2 (0.43) ADRB2CNR2LDHALDHBLMNA
SCHEMBL681142 0.82 KMT2A (0.42) ADRB2LMNACYP1A2CYP2D6TSHR
SCHEMBL681371 0.82 KMT2A (0.42) ADRB2LMNACYP1A2CYP2D6TSHR
SCHEMBL681782 0.82 CYP1A2 (0.38) ADRB2LMNACYP1A2CYP2D6TSHR
SCHEMBL681368 0.82 KMT2A (0.42) ADRB2LMNACYP1A2CYP2D6TSHR
SCHEMBL2738443 0.81 CNR2 (0.45) ADRB2CNR2LDHALDHBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8063050-B2 Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors ARRAY BIOPHARMA INC. (US) 2011-11-22 US disclosed