SCHEMBL681564

SCHEMBL681564

C=C(C(C)C)C(CNC(C)C)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
PSEN1 P49768 1/20 0.37
PSEN2 P49810 1/20 0.37
APH1B Q8WW43 1/20 0.37
NCSTN Q92542 1/20 0.37
APH1A Q96BI3 1/20 0.37
PSENEN Q9NZ42 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
CNR2 P34972 1/20 0.36
TEAD1 P28347 2/20 0.36
LDHA P00338 2/20 0.36
LDHB P07195 2/20 0.36
CYP3A4 P08684 1/20 0.36
PDE2A O00408 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL681594 1.00 CA1 (0.38) CA1CA2PSEN1PSEN2APH1B
SCHEMBL681195 0.85 PSEN1 (0.40) CA1CA2PSEN1PSEN2APH1B
SCHEMBL679682 0.85 PSEN1 (0.40) CA1CA2PSEN1PSEN2APH1B
SCHEMBL681163 0.85 TACR1 (0.37) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL681259 0.84 ADRB2 (0.40) CA1CA2PSEN1PSEN2APH1B
SCHEMBL684568 0.84 PSEN1 (0.41) CA1CA2PSEN1PSEN2APH1B
SCHEMBL12188333 0.84 PSEN1 (0.41) CA1CA2PSEN1PSEN2APH1B
SCHEMBL680060 0.83 ADRB2 (0.44) ALDH1A1CYP3A4
SCHEMBL2738579 0.82 CNR2 (0.42) CA1CA2PSEN1PSEN2APH1B
SCHEMBL2738513 0.82 CNR2 (0.42) CA1CA2PSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8063050-B2 Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors ARRAY BIOPHARMA INC. (US) 2011-11-22 US disclosed