SCHEMBL6816154

SCHEMBL6816154

CC(C)(C)C[C@@H](N)C(=O)NC(=O)C1C[C@@H](F)CN1Cc1cc(Cl)ccc1-c1cnccn1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 2/20 0.36
P2RX7 Q99572 2/20 0.33
PTGES2 Q9H7Z7 1/20 0.33
GRM5 P41594 1/20 0.32
MAOA P21397 2/20 0.32
MAOB P27338 2/20 0.32
AAK1 Q2M2I8 2/20 0.32
CIT O14578 1/20 0.31
HIPK4 Q8NE63 1/20 0.31
MKNK2 Q9HBH9 1/20 0.31
BMP2K Q9NSY1 1/20 0.31
KMT2A Q03164 1/20 0.31
DPP4 P27487 1/20 0.31
TRPA1 O75762 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6819766 0.81 MAOB (0.45) GPBAR1P2RX7PTGES2GRM5MAOA
SCHEMBL6921204 0.80 F2 (0.40) GPBAR1AAK1KMT2A
SCHEMBL6916861 0.78 CYP3A4 (0.45) GPBAR1
SCHEMBL6921736 0.78 CYP3A4 (0.45) GPBAR1
SCHEMBL6919934 0.78 CYP3A4 (0.45) GPBAR1
SCHEMBL6918997 0.78 CYP3A4 (0.45) GPBAR1
SCHEMBL6918706 0.77 GPBAR1 (0.36) GPBAR1MAOAMAOBDPP4
SCHEMBL6914935 0.71 GPBAR1 (0.34) GPBAR1AAK1TRPA1
SCHEMBL6921239 0.70 F2 (0.38) GPBAR1AAK1KMT2A
SCHEMBL6922183 0.69 CYP3A4 (0.48) GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004032834-A2 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2004-04-22 WO claimed