SCHEMBL6914935

SCHEMBL6914935

CC(C)(C)OC(=O)N[C@@H](C(=O)NC(=O)[C@@H]1C[C@@H](F)CN1Cc1cc(Cl)ccc1-c1cnsn1)C(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 2/20 0.34
CTRB1 P17538 2/20 0.32
PTGER1 P34995 1/20 0.32
ENPP2 Q13822 1/20 0.31
TRPA1 O75762 1/20 0.31
AAK1 Q2M2I8 1/20 0.30
SCN9A Q15858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6918706 0.87 GPBAR1 (0.36) GPBAR1
SCHEMBL6914941 0.82 VHL (0.38)
SCHEMBL6816154 0.71 GPBAR1 (0.36) GPBAR1TRPA1AAK1
SCHEMBL6918709 0.71 F2 (0.41)
SCHEMBL6919609 0.69 CFD (0.40) TRPA1
SCHEMBL6920452 0.68 SCN9A (0.36) GPBAR1AAK1SCN9A
SCHEMBL6919273 0.67 SCN9A (0.35) GPBAR1PTGER1ENPP2AAK1SCN9A
SCHEMBL6078132 0.67 F2 (0.51)
SCHEMBL6921239 0.65 F2 (0.38) GPBAR1AAK1
SCHEMBL6922183 0.65 CYP3A4 (0.48) GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004032834-A2 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2004-04-22 WO disclosed