SCHEMBL6818176

SCHEMBL6818176

CN(C)c1cc(Cl)c(-c2ccnc(NCCCC3CC3)c2[N+](=O)[O-])cc1F

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 2/20 0.33
NPC1 O15118 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
CASP3 P42574 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
SENP8 Q96LD8 1/20 0.33
SENP7 Q9BQF6 1/20 0.33
SENP6 Q9GZR1 1/20 0.33
CCR2 P41597 2/20 0.32
KCNH2 Q12809 1/20 0.32
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
CYP2C9 P11712 1/20 0.30
PRKCQ Q04759 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6822478 0.95 CYP3A4 (0.33) MAPTCYP3A4CYP2D6NPC1CYP1A2
SCHEMBL6813930 0.86 SCN9A (0.37) MAPTCYP3A4CYP2D6NPC1CYP1A2
SCHEMBL6814158 0.85 ALDH1A1 (0.33) MAPTCYP3A4CYP2D6NPC1CYP1A2
SCHEMBL6814612 0.84 BCHE (0.30)
SCHEMBL6817813 0.82 PRKCQ (0.39) MAPTCYP3A4CYP2D6NPC1CYP1A2
SCHEMBL6817921 0.80 MAPT (0.36) MAPTNPC1SMN1; SMN2KCNH2MEN1
SCHEMBL6821721 0.80 NPC1 (0.34) MAPTNPC1RAB9ASMN1; SMN2KCNH2
SCHEMBL6814129 0.80 PRKCQ (0.38) MAPTCYP3A4CYP2D6NPC1CYP1A2
SCHEMBL6082249 0.79 IDH1 (0.36) CYP2C19CYP2C9
SCHEMBL6082255 0.79 IDH1 (0.36) CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004031189-A1 PYRIDINO AND PYRIMIDINO PYRAZINONES FOR TREATMENT OF ANXIETY AND DEPRESSION BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2004-04-15 WO disclosed