SCHEMBL6818256

SCHEMBL6818256

COC(=O)Cc1ccc2oc(-c3ccc([N+](=O)[O-])c(C)c3)nc2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.58
ALDH1A1 P00352 2/20 0.58
KDM4E B2RXH2 1/20 0.58
MAPK1 P28482 1/20 0.58
MAPT P10636 6/20 0.50
TP53 P04637 3/20 0.50
THRB P10828 2/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
SLC2A1 P11166 1/20 0.48
HPSE Q9Y251 3/20 0.47
RAB9A P51151 3/20 0.47
MMP2 P08253 1/20 0.46
MMP9 P14780 1/20 0.46
MMP8 P22894 1/20 0.46
MMP13 P45452 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
PPARG P37231 1/20 0.45
CETP P11597 1/20 0.45
CEPT1 Q9Y6K0 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6824973 0.89 NPC1 (0.57) NPC1ALDH1A1KDM4EMAPK1MAPT
SCHEMBL6822112 0.87 NPC1 (0.57) NPC1ALDH1A1KDM4EMAPK1MAPT
SCHEMBL6821886 0.85 NPC1 (0.62) NPC1ALDH1A1KDM4EMAPK1MAPT
SCHEMBL6821781 0.83 NPC1 (0.62) NPC1ALDH1A1KDM4EMAPK1MAPT
SCHEMBL6821840 0.83 NPC1 (0.65) NPC1ALDH1A1KDM4EMAPK1MAPT
SCHEMBL6822046 0.82 NPC1 (0.58) NPC1ALDH1A1KDM4EMAPK1MAPT
Methane SCHEMBL6821779 0.81 NPC1 (0.57) NPC1ALDH1A1KDM4EMAPK1MAPT
SCHEMBL5465423 0.79 PDGFRB (0.53) NPC1ALDH1A1MAPK1MAPTMEN1
SCHEMBL6818285 0.79 NPC1 (0.67) NPC1ALDH1A1KDM4EMAPK1MAPT
SCHEMBL6821837 0.79 NPC1 (0.67) NPC1ALDH1A1KDM4EMAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004046122-A2 BENZOXAZOLE, BENZTHIAZOLE AND BENZIMIDAZOLE ACID DERIVATIVES AND THEIR USE AS HEPARANASE INHIBITORS OXFORD GLYCOSCIENCES (UK) LTD (GB) 2004-06-03 WO disclosed