SCHEMBL6818583

SCHEMBL6818583

CC(=O)Nc1ccc(-c2cc3onc(C(=O)Nc4ccc(C#N)cc4C(=O)O)c3cc2C(=O)N(C)C)c(C(F)(F)F)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.33
TP53 P04637 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
MAP2K1 Q02750 1/20 0.33
S1PR1 P21453 2/20 0.32
S1PR3 Q99500 2/20 0.32
ALB P02768 2/20 0.32
TAS2R14 Q9NYV8 1/20 0.31
HIF1A Q16665 1/20 0.31
MPO P05164 1/20 0.31
RAPGEF3 O95398 2/20 0.31
RAPGEF4 Q8WZA2 1/20 0.31
F10 P00742 1/20 0.31
APP P05067 1/20 0.31
CTSD P07339 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
BACE1 P56817 1/20 0.31
BACE2 Q9Y5Z0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6821658 0.98 RORC (0.33) RORCTP53POLBMAPTMAP2K1
SCHEMBL6819217 0.91 PDE10A (0.37) RORCTP53POLBMAPTMAP2K1
SCHEMBL6818406 0.91 RORC (0.34) RORCTP53POLBMAPTMAP2K1
SCHEMBL6833954 0.90 RORC (0.35) RORCTP53POLBMAPTMAP2K1
SCHEMBL6822026 0.90 EGLN2 (0.35) RORCTP53POLBMAPTMAP2K1
SCHEMBL6818615 0.89 RORC (0.35) RORCMAP2K1S1PR1S1PR3ALB
SCHEMBL6818625 0.89 MAP2K1 (0.34) RORCTP53POLBMAPTMAP2K1
SCHEMBL6818778 0.89 PDE10A (0.37) RORCTP53POLBMAPTMAP2K1
SCHEMBL6818889 0.89 EGLN2 (0.34) RORCTP53POLBMAPTMAP2K1
SCHEMBL6813970 0.89 TP53 (0.35) TP53ALBHIF1AF10RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004018428-A1 ANTIBACTERIAL BENZOIC ACID DERIVATIVES PHARMACIA & UPJOHN COMPANY LLC (US) 2004-03-04 WO disclosed