SCHEMBL6823205

SCHEMBL6823205

CNc1nc2sc(-c3cccc(CC(C)NC(C)=O)c3)nc2c2c1ncn2C

nearest known ligand 0.77

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 20/20 0.77
CHUK O15111 9/20 0.77
CDK2 P24941 1/20 0.75
BTK Q06187 1/20 0.75
ITK Q08881 1/20 0.75
IKBKE Q14164 1/20 0.75
JAK2 O60674 1/20 0.59
TYK2 P29597 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5659332 0.87 IKBKB (1.00) IKBKBCHUKCDK2BTKITK
SCHEMBL6826475 0.87 IKBKB (0.70) IKBKBCHUKCDK2BTKITK
SCHEMBL5657326 0.86 IKBKB (1.00) IKBKBCHUKCDK2BTKITK
SCHEMBL6823454 0.85 IKBKB (0.85) IKBKBCHUKCDK2BTKITK
SCHEMBL5657089 0.82 IKBKB (0.74) IKBKBCHUKCDK2BTKITK
SCHEMBL14589256 0.81 IKBKB (0.72) IKBKBCHUKCDK2BTKITK
SCHEMBL16794616 0.80 IKBKB (0.72) IKBKBCHUKCDK2BTKITK
SCHEMBL6823062 0.80 IKBKB (0.72) IKBKBCHUKCDK2BTKITK
SCHEMBL14589469 0.79 IKBKB (0.70) IKBKBCHUKCDK2BTKITK
SCHEMBL14589410 0.79 IKBKB (0.74) IKBKBCHUKCDK2BTKITK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004106293-A2 OXAZOLYL - AND THIAZOLYL - PURINE BASED TRICYCLIC COMPOUNDS. BRISTOL-MYERS SQUIBB COMPANY (US) 2004-12-09 WO claimed