SCHEMBL6823372

SCHEMBL6823372

c1ccc2c(Nc3ccncc3)ncnc2c1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 8/20 0.77
ABCG2 Q9UNQ0 5/20 0.77
ERBB2 P04626 2/20 0.77
AURKB Q96GD4 2/20 0.77
CLK4 Q9HAZ1 2/20 0.77
DAPK3 O43293 1/20 0.77
MAP4K4 O95819 1/20 0.77
ABL1 P00519 1/20 0.77
PIM1 P11309 1/20 0.77
PRKACA P17612 1/20 0.77
LTK P29376 1/20 0.77
MAPK8 P45983 1/20 0.77
CSNK1A1 P48729 1/20 0.77
RPS6KA3 P51812 1/20 0.77
LIMK1 P53667 1/20 0.77
MAP2K1 Q02750 1/20 0.77
ACVR1 Q04771 1/20 0.77
TYRO3 Q06418 1/20 0.77
MAP4K2 Q12851 1/20 0.77
ROCK1 Q13464 1/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29941271 0.87 EGFR (1.00) EGFRABCG2ERBB2AURKBCLK4
SCHEMBL8920 0.87 EGFR (1.00) EGFRABCG2ERBB2AURKBCLK4
Hydrochloric Acid SCHEMBL20856873 0.86 EGFR (0.96) EGFRABCG2ERBB2AURKBCLK4
Hydrochloric Acid SCHEMBL29394578 0.86 EGFR (0.96) EGFRABCG2ERBB2AURKBCLK4
SCHEMBL8976752 0.83 EGFR (0.78) EGFRABCG2ERBB2AURKBCLK4
SCHEMBL31375768 0.83 EGFR (0.65) EGFRABCG2ERBB2AURKBCLK4
Hydrochloric Acid SCHEMBL8808235 0.83 EGFR (0.90) EGFRABCG2ERBB2AURKBCLK4
SCHEMBL6823152 0.82 EGFR (0.71) EGFRABCG2ERBB2AURKBCLK4
SCHEMBL14027230 0.81 EGFR (0.75) EGFRABCG2ERBB2AURKBCLK4
SCHEMBL5569041 0.81 EGFR (0.75) EGFRABCG2ERBB2AURKBCLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023081800-A1 ALPHA-2A ADRENERGIC RECEPTOR MODULATORS AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-05-11 WO disclosed
WO-2004056812-A1 4- (PYRIDIN-4-YLAMINO) -QUINAZOLINE DERIVATIVES AS ANTI-TUMOR AGENTS ASTRAZENECA AB (SE) 2004-07-08 WO disclosed