SCHEMBL6824480

SCHEMBL6824480

COC(=O)c1ccc(C2=CCNC(C(=O)OC(C)(C)C)C2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 3/20 0.38
F2 P00734 1/20 0.37
CA1 P00915 4/20 0.36
CA2 P00918 4/20 0.36
CA12 O43570 3/20 0.36
CA9 Q16790 3/20 0.36
CA14 Q9ULX7 3/20 0.36
TDP1 Q9NUW8 1/20 0.36
CA7 P43166 1/20 0.36
HTT P42858 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
RECQL P46063 1/20 0.35
EGFR P00533 1/20 0.35
WNT3A P56704 1/20 0.35
TNKS2 Q9H2K2 1/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
NOTUM Q6P988 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4427892 0.82 CRBN (0.34) KDM4EKMT2ARECQL
SCHEMBL7261773 0.81 CYP11B1 (0.38) KDM4EALDH1A1F2TDP1HTT
SCHEMBL7527330 0.80 MAPT (0.41) ALDH1A1HTTMEN1KMT2AGAA
SCHEMBL6647089 0.78 MIF (0.34) HDAC1HDAC6
SCHEMBL3657554 0.75 F2 (0.33) F2
SCHEMBL6829492 0.75 F2 (0.35) F2
SCHEMBL4441491 0.74 RECQL (0.33) RECQL
SCHEMBL6648198 0.74 NQO2 (0.43) KDM4EALDH1A1MEN1KMT2AHPGD
SCHEMBL7510927 0.72 MIF (0.43) HDAC6
SCHEMBL27387819 0.72 HTT (0.43) KDM4EALDH1A1CA1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004058727-A1 SUBSTITUTED 3,5-DIHYDRO-4H-IMIDAZOL-4-ONES FOR THE TREATMENT OF OBESITY BAYER PHARMACEUTICALS CORPORATION (US) 2004-07-15 WO disclosed