SCHEMBL6824968

SCHEMBL6824968

COc1ccc2c(c1)c(=O)oc1c(C)c(O)ccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 14/20 1.00
ESR1 P03372 10/20 0.69
HSD17B10 Q99714 1/20 0.61
POLB P06746 4/20 0.59
MAPT P10636 2/20 0.58
KDM4E B2RXH2 1/20 0.57
NPC1 O15118 1/20 0.57
ALDH1A1 P00352 1/20 0.57
STAT1 P42224 1/20 0.57
RAB9A P51151 1/20 0.57
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
CTDSP1 Q9GZU7 2/20 0.56
PKM P14618 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29853599 0.84 ESR2 (0.73) ESR2ESR1HSD17B10POLBMAPT
SCHEMBL26766950 0.84 ESR2 (0.73) ESR2ESR1HSD17B10POLBMAPT
SCHEMBL12813762 0.84 ESR2 (0.72) ESR2ESR1HSD17B10POLBMAPT
SCHEMBL11843906 0.82 ESR2 (0.70) ESR2ESR1HSD17B10POLBMAPT
SCHEMBL6828078 0.82 ESR2 (1.00) ESR2ESR1KDM4EALDH1A1
SCHEMBL6825648 0.82 ESR2 (0.77) ESR2ESR1KDM4EALDH1A1
SCHEMBL22413028 0.81 ESR2 (0.77) ESR2ESR1
SCHEMBL6825403 0.79 ESR2 (1.00) ESR2ESR1KDM4EALDH1A1
SCHEMBL6828126 0.79 ESR2 (0.73) ESR2ESR1KDM4EALDH1A1
SCHEMBL29853560 0.79 KDM4E (0.79) ESR2ESR1HSD17B10POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004073612-A2 ESTROGEN RECEPTOR MODULATORS MERCK & CO. INC. (US) 2004-09-02 WO claimed
EP-2691542-A1 SCREENING METHODS FOR IDENTIFYING SPECIFIC STAPHYLOCOCCUS AUREUS INHIBITORS Trana Discovery, Inc. (US) 2014-02-05 EP disclosed
WO-2012135416-A1 SCREENING METHODS FOR IDENTIFYING SPECIFIC STAPHYLOCOCCUS AUREUS INHIBITORS TRANA DISCOVERY, INC. (US) 2012-10-04 WO disclosed
WO-2004073612-A2 ESTROGEN RECEPTOR MODULATORS MERCK & CO. INC. (US) 2004-09-02 WO disclosed