SCHEMBL6825503

SCHEMBL6825503

O=C(O)CC1COC2(CCN(Cc3ccccc3)CC2)C1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 2/20 0.54
FFAR1 O14842 2/20 0.51
CYP2D6 P10635 3/20 0.50
SIGMAR1 Q99720 5/20 0.49
TMEM97 Q5BJF2 2/20 0.49
OPRM1 P35372 1/20 0.47
ALDH1A1 P00352 2/20 0.46
CYP3A4 P08684 2/20 0.46
USP2 O75604 1/20 0.46
MAPK1 P28482 1/20 0.46
CHRM2 P08172 3/20 0.46
CHRM3 P20309 2/20 0.46
OPRL1 P41146 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6823088 0.81 SIGMAR1 (0.50) FFAR1CYP2D6SIGMAR1TMEM97OPRM1
SCHEMBL6819672 0.77 SIGMAR1 (0.47) CYP2D6SIGMAR1TMEM97CHRM2CHRM3
SCHEMBL6747206 0.76 CXCR4 (0.65)
Hydrochloric Acid SCHEMBL9537230 0.75 BCHE (0.63)
SCHEMBL1966477 0.74 SIGMAR1 (0.61) CYP2D6SIGMAR1TMEM97OPRM1ALDH1A1
SCHEMBL21590941 0.74 FFAR1 (0.50) FFAR1CYP2D6SIGMAR1TMEM97OPRM1
SCHEMBL2524338 0.73 CYP2D6 (0.57) CYP2D6SIGMAR1ALDH1A1CYP3A4USP2
SCHEMBL4023771 0.72 OPRL1 (0.59) CYP2D6SIGMAR1ALDH1A1CYP3A4USP2
Hydrochloric Acid SCHEMBL4481783 0.72 POLB (0.58) CYP2D6SIGMAR1ALDH1A1CYP3A4USP2
SCHEMBL21590851 0.71 SIGMAR1 (0.48) FFAR1SIGMAR1TMEM97OPRM1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004058763-A1 4(SPIROPIPERIDINYL)METHYL SUBSTITUTED PYRROLIDINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 2004-07-15 WO disclosed