SCHEMBL6825854

SCHEMBL6825854

Cn1nc(C(N)=O)cc1C#N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G10 O15496 3/20 0.44
L3MBTL1 Q9Y468 1/20 0.40
BAZ2B Q9UIF8 1/20 0.39
LRRK2 Q5S007 1/20 0.38
GSK3B P49841 1/20 0.36
FAAH O00519 1/20 0.34
PIM3 Q86V86 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
LMNA P02545 1/20 0.33
GRM2 Q14416 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
SCN9A Q15858 2/20 0.32
MYC P01106 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16468110 0.84 BAZ2B (0.40) L3MBTL1BAZ2BLRRK2KDM4EALDH1A1
SCHEMBL6826183 0.79 AR (0.41) BAZ2BLRRK2LMNAKDM4EALDH1A1
SCHEMBL31739403 0.79 MALT1 (0.38) BAZ2BLRRK2KDM4EALDH1A1
SCHEMBL4751927 0.77 PLA2G10 (0.49) PLA2G10L3MBTL1BAZ2BGSK3BFAAH
SCHEMBL1080282 0.77 BAZ2B (0.61) PLA2G10L3MBTL1BAZ2BGSK3BPIM3
SCHEMBL24914934 0.76 GAA (0.43) L3MBTL1FAAHLMNAKDM4EALDH1A1
Hydrochloric Acid SCHEMBL3491832 0.76 BAZ2B (0.59) PLA2G10L3MBTL1BAZ2BGSK3BPIM3
SCHEMBL29092152 0.73 PLA2G10 (0.49) PLA2G10L3MBTL1BAZ2BGSK3BFAAH
SCHEMBL15942241 0.73 PLA2G10 (0.49) PLA2G10L3MBTL1BAZ2BGSK3BFAAH
SCHEMBL29080123 0.72 PLA2G10 (0.47) PLA2G10L3MBTL1BAZ2BGSK3BFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6740647-B1 AMIDINES AND HYDROXYAMIDINE DERIVATIVES ABBOTT GMBH & CO., KG (DE) 2004-05-25 US disclosed
CN-1289341-A Thrombin inhibitors BASF AG (DE) 2001-03-28 CN disclosed
CN-1228783-A Novel thrombin inhibitors BASF AG (DE) 1999-09-15 CN disclosed