SCHEMBL6828068

SCHEMBL6828068

COc1c(C)c(Br)c(CO)c(Br)c1C

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA2 P00918 10/20 0.65
CA4 P22748 6/20 0.65
CA1 P00915 8/20 0.41
CA6 P23280 4/20 0.41
DRD4 P21917 1/20 0.39
PTPN1 P18031 1/20 0.35
IMPDH2 P12268 3/20 0.33
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
CA12 O43570 3/20 0.31
CA9 Q16790 2/20 0.31
AKR1B1 P15121 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15961197 0.79 CA2 (1.00) CA2CA4CA1CA6DRD4
SCHEMBL6828106 0.78 CA2 (0.50) CA2CA4CA1CA6PTPN1
SCHEMBL22402725 0.78 DRD4 (0.48) CA2CA4DRD4
SCHEMBL9549629 0.76 CA2 (0.46) CA2CA4IMPDH2AKR1B1
SCHEMBL6825433 0.73 DRD4 (0.56) CA2CA4CA1CA6DRD4
SCHEMBL11389950 0.72 DRD4 (0.55) CA2CA4CA1CA6DRD4
SCHEMBL1783863 0.72 CA2 (0.39) CA2CA4CA1CA6PTPN1
SCHEMBL14946904 0.72 CA2 (0.39) CA2CA4CA1CA6PTPN1
SCHEMBL9070629 0.72 CA2 (0.42) CA2CA4CA1CA6PTPN1
SCHEMBL7971157 0.71 CA2 (0.46) CA2CA4CA1CA6IMPDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004073612-A2 ESTROGEN RECEPTOR MODULATORS MERCK & CO. INC. (US) 2004-09-02 WO disclosed