SCHEMBL6828569

SCHEMBL6828569

O=S(=O)(Nc1ccccc1)c1ccc2[nH]c3c(Cl)ncnc3c2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 3/20 0.54
PKM P14618 1/20 0.53
KDM4E B2RXH2 3/20 0.52
MAPT P10636 3/20 0.52
ALDH1A1 P00352 3/20 0.52
MAPK1 P28482 1/20 0.52
POLB P06746 1/20 0.49
PDE3A Q14432 1/20 0.47
PGR P06401 1/20 0.44
PLG P00747 1/20 0.43
PLAU P00749 1/20 0.43
PLAT P00750 1/20 0.43
LMNA P02545 2/20 0.43
TP53 P04637 1/20 0.43
THRB P10828 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
BRD4 O60885 2/20 0.42
EGFR P00533 1/20 0.42
HTR2C P28335 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6822894 0.84 POLB (0.55) PKMKDM4EMAPTALDH1A1MAPK1
SCHEMBL6828688 0.80 KDM4E (0.62) BRAFKDM4EMAPTALDH1A1MAPK1
SCHEMBL6826630 0.79 KDM4E (0.60) BRAFKDM4EMAPTALDH1A1MAPK1
SCHEMBL6826652 0.74 ABCB1 (0.54) KDM4EMAPTALDH1A1MAPK1POLB
SCHEMBL31219113 0.72 KDM4E (0.72) KDM4EMAPTALDH1A1MAPK1POLB
SCHEMBL17396514 0.72 KDM4E (0.72) KDM4EMAPTALDH1A1MAPK1POLB
SCHEMBL6254106 0.71 LIMK1 (0.65) KDM4EMAPTALDH1A1MAPK1POLB
SCHEMBL6826964 0.71 KDM4E (0.50) KDM4EMAPTALDH1A1MAPK1POLB
SCHEMBL27829906 0.70 BRAF (1.00) BRAFPKMPDE3APLGPLAU
Hydrochloric Acid SCHEMBL7221411 0.70 LIMK1 (0.63) KDM4EMAPTALDH1A1MAPK1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004111052-A1 PYRROLOPYRIMIDINE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE (MDR) XENOVA LIMITED (GB) 2004-12-23 WO disclosed