SCHEMBL6828937

SCHEMBL6828937

Cc1cc2c(c(C)c1NC(=O)N1CCCC(C(=O)O)C1)c1ccccc1n2C(C)C

nearest known ligand 0.67

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 7/20 0.67
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HTT P42858 1/20 0.42
CREBBP Q92793 1/20 0.41
HPGD P15428 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
SHMT2 P34897 1/20 0.39
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6829275 0.95 NPY5R (0.69) NPY5RKMT2AHTTMAPTALDH1A1
SCHEMBL6823362 0.92 NPY5R (0.66) NPY5RKMT2AKDM4EHSD17B10HTT
SCHEMBL6826749 0.91 NPY5R (0.65) NPY5RKMT2AKDM4EHSD17B10HTT
SCHEMBL6826597 0.91 NPY5R (0.64) NPY5RKMT2AKDM4EHSD17B10HTT
SCHEMBL6823308 0.89 NPY5R (0.62) NPY5RKMT2AHTTHPGDGAA
SCHEMBL6826590 0.88 NPY5R (0.60) NPY5RKMT2AKDM4EHSD17B10GAA
SCHEMBL7087839 0.86 NPY5R (0.58) NPY5RKMT2AKDM4EHSD17B10HTT
SCHEMBL6826986 0.86 NPY5R (0.67) NPY5RKDM4EHTTCREBBPGAA
SCHEMBL6827520 0.85 NPY5R (0.66) NPY5RKMT2AKDM4EHSD17B10HTT
SCHEMBL6829075 0.85 NPY5R (0.66) NPY5RKMT2AKDM4EHSD17B10HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040067999-A1 Carbazole derivatives and their use as neuropeptide y5 receptor ligands ASTRAZENECA AB (SE) 2004-04-08 US disclosed
EP-1358157-A1 CARBAZOLE DERIVATIVES AND THEIR USE AS NEUROPEPTIDE Y5 RECEPTOR LIGANDS AstraZeneca AB (SE) 2003-11-05 EP disclosed
WO-2002051806-A1 CARBAZOLE DERIVATIVES AND THEIR USE AS NEUROPEPTIDE Y5 RECEPTOR LIGANDS ASTRAZENECA AB (SE) 2002-07-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040067999-A1 Carbazole derivatives and their use as neuropeptide y5 receptor ligands NPY5R, NPY1R, NPY2R NPY5R 1/4885KMT2A 3618/4885KDM4E 2632/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.