SCHEMBL7087839

SCHEMBL7087839

Cc1cc2c(c(C)c1NC(=O)C(Cl)(Cl)Cl)c1ccccc1n2C(C)C.Cc1cc2c(c(C)c1NC(=O)N1CCCC(C(N)=O)C1)c1ccccc1n2C(C)C

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 7/20 0.58
KDM4E B2RXH2 2/20 0.47
HSD17B10 Q99714 1/20 0.47
LMNA P02545 1/20 0.37
KMT2A Q03164 2/20 0.37
RAB9A P51151 1/20 0.36
HTT P42858 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
SHMT2 P34897 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6823362 0.94 NPY5R (0.66) NPY5RKDM4EHSD17B10LMNAKMT2A
SCHEMBL6828937 0.86 NPY5R (0.67) NPY5RKDM4EHSD17B10KMT2AHTT
SCHEMBL6826749 0.85 NPY5R (0.65) NPY5RKDM4EHSD17B10LMNAKMT2A
SCHEMBL6826597 0.84 NPY5R (0.64) NPY5RKDM4EHSD17B10LMNAKMT2A
SCHEMBL6823308 0.83 NPY5R (0.62) NPY5RLMNAKMT2ARAB9AHTT
SCHEMBL6823236 0.82 NPY5R (0.63) NPY5RKDM4EKMT2AHTTGAA
SCHEMBL6826590 0.81 NPY5R (0.60) NPY5RKDM4EHSD17B10KMT2ARAB9A
SCHEMBL6829275 0.81 NPY5R (0.69) NPY5RKMT2ARAB9AHTTMAPT
SCHEMBL6826741 0.80 NPY5R (0.65) NPY5RKDM4EHSD17B10LMNAKMT2A
SCHEMBL6826986 0.80 NPY5R (0.67) NPY5RKDM4ERAB9AHTTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1358157-A1 CARBAZOLE DERIVATIVES AND THEIR USE AS NEUROPEPTIDE Y5 RECEPTOR LIGANDS AstraZeneca AB (SE) 2003-11-05 EP disclosed
WO-2002051806-A1 CARBAZOLE DERIVATIVES AND THEIR USE AS NEUROPEPTIDE Y5 RECEPTOR LIGANDS ASTRAZENECA AB (SE) 2002-07-04 WO disclosed