SCHEMBL6829077

SCHEMBL6829077

Cc1cc2c(c(C)c1NC(=O)C1CCNCC1)c1ccccc1n2C(C)C

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 8/20 0.61
HTR4 Q13639 6/20 0.41
KHK P50053 1/20 0.39
KCNH2 Q12809 1/20 0.39
TP53 P04637 2/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
GNRHR P30968 1/20 0.37
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6829078 0.87 NPY5R (0.63) NPY5RTP53LMNAMAPTPOLB
SCHEMBL6823457 0.86 NPY5R (0.62) NPY5RTP53LMNAMAPTPOLB
SCHEMBL6828992 0.86 NPY5R (0.67) NPY5RMAPT
SCHEMBL6823387 0.85 NPY5R (0.61) NPY5RTP53LMNAMAPT
SCHEMBL6826862 0.84 NPY5R (0.61) NPY5RTP53LMNAMAPTPOLB
SCHEMBL6824384 0.82 NPY5R (0.59) NPY5RTP53LMNAMAPT
SCHEMBL6823480 0.81 NPY5R (0.56) NPY5R
SCHEMBL6826590 0.81 NPY5R (0.60) NPY5RMAPTPOLB
SCHEMBL6823236 0.80 NPY5R (0.63) NPY5RMAPTPOLB
SCHEMBL6990117 0.79 NPY5R (0.44) NPY5RHTR4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1531527-A Carbazole derivatives and their use as neuropeptide Y5 receptor ligands 2004-09-22 CN disclosed
US-20040067999-A1 Carbazole derivatives and their use as neuropeptide y5 receptor ligands ASTRAZENECA AB (SE) 2004-04-08 US disclosed
EP-1358157-A1 CARBAZOLE DERIVATIVES AND THEIR USE AS NEUROPEPTIDE Y5 RECEPTOR LIGANDS AstraZeneca AB (SE) 2003-11-05 EP disclosed
WO-2002051806-A1 CARBAZOLE DERIVATIVES AND THEIR USE AS NEUROPEPTIDE Y5 RECEPTOR LIGANDS ASTRAZENECA AB (SE) 2002-07-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040067999-A1 Carbazole derivatives and their use as neuropeptide y5 receptor ligands NPY5R, NPY1R, NPY2R NPY5R 1/4885HTR4 136/4885KHK 2546/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.