SCHEMBL6829462

SCHEMBL6829462

Fc1ccccc1C=CBr

nearest known ligand 0.75

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 13/20 0.75
RELA Q04206 2/20 0.47
NPC1 O15118 1/20 0.46
PKM P14618 1/20 0.46
NFKB1 P19838 1/20 0.46
RAB9A P51151 1/20 0.46
NFKB2 Q00653 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MAOB P27338 1/20 0.44
GRM4 Q14833 1/20 0.43
GRIN2D O15399 1/20 0.42
GRIN3B O60391 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42
GRIN2C Q14957 1/20 0.42
GRIN3A Q8TCU5 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL38650720 1.00 NFE2L2 (0.75) NFE2L2RELANPC1PKMNFKB1
SCHEMBL2234105 0.86 NFE2L2 (1.00) NFE2L2RELANPC1PKMNFKB1
SCHEMBL15353049 0.81
SCHEMBL11209913 0.80 NFE2L2 (0.43) NFE2L2NFKB1MAOB
SCHEMBL575116 0.78
SCHEMBL14162953 0.77 NFE2L2 (0.71) NFE2L2RELANPC1PKMNFKB1
SCHEMBL6804693 0.77 NFE2L2 (0.71) NFE2L2RELANPC1PKMNFKB1
SCHEMBL2089367 0.77 NFE2L2 (0.71) NFE2L2RELANPC1PKMNFKB1
SCHEMBL2089369 0.77 NFE2L2 (0.71) NFE2L2RELANPC1PKMNFKB1
SCHEMBL3434176 0.77 NFE2L2 (0.71) NFE2L2RELANPC1PKMNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113511972-A (E) Preparation method of (E) -4-aryl-2, 2-difluoro-3-butenoic acid derivative 昆明理工大学 2021-10-19 CN disclosed
CN-100389113-C Nitrogen-containing heterocyclic compound and drug containing same EISAI CO LTD (JP) 2008-05-21 CN disclosed
CN-1630650-A Nitrogen-containing heterocyclic compound and drug containing same EISAI CO LTD (JP) 2005-06-22 CN disclosed
EP-1159265-B1 C-16 UNSATURATED FP-SELECTIVE PROSTAGLANDINS ANALOGS UNIV DUKE (US) 2004-11-24 EP disclosed
US-6451859-B1 C16 unsaturated FP-selective prostaglandins analogs THE PROCTER & GAMBLE COMPANY 2002-09-17 US disclosed
EP-1159265-A1 C-16 UNSATURATED FP-SELECTIVE PROSTAGLANDINS ANALOGS THE PROCTER & GAMBLE COMPANY (US) 2001-12-05 EP disclosed
WO-2000051979-A1 C16 UNSATURATED FP-SELECTIVE PROSTAGLANDINS ANALOGS THE PROCTER & GAMBLE COMPANY (US) 2000-09-08 WO disclosed