SCHEMBL6829600

SCHEMBL6829600

CSc1cc(C)nc(N)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 3/20 0.49
TSHR P16473 4/20 0.47
CYP1A2 P05177 2/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HSP90AA1 P07900 1/20 0.45
LMNA P02545 3/20 0.45
MAPT P10636 2/20 0.45
NPC1 O15118 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
GAA P10253 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.40
CRHBP P24387 1/20 0.40
CRHR2 Q13324 1/20 0.40
CYP2D6 P10635 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
NUDT1 P36639 1/20 0.39
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28486478 0.84 HSP90AB1 (0.50) HSP90AB1TSHRCYP1A2HSP90AA1LMNA
SCHEMBL741180 0.84 HSP90AB1 (0.50) HSP90AB1TSHRCYP1A2HSP90AA1LMNA
SCHEMBL763785 0.79 HRH4 (0.37) HSP90AB1HSP90AA1MAPTNPC1HRH3
SCHEMBL151114 0.77
SCHEMBL13744682 0.77 TSHR (0.59) HSP90AB1TSHRCYP1A2HSP90AA1LMNA
SCHEMBL21711151 0.76 CYP1A2 (0.48) HSP90AB1CYP1A2CYP2C9CYP2C19LMNA
SCHEMBL191457 0.76 KMT2A (0.59) HSP90AB1CYP1A2CYP2C19HSP90AA1LMNA
SCHEMBL7568606 0.75 HSP90AB1 (0.55) HSP90AB1TSHRCYP1A2HSP90AA1LMNA
SCHEMBL7568049 0.75 HSP90AB1 (0.55) HSP90AB1TSHRCYP1A2CYP2C19HSP90AA1
Ammonia Solution, Strong SCHEMBL20919221 0.75 HSP90AA1 (0.56) HSP90AB1TSHRCYP1A2CYP2C19HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1463483-A1 NEW COMPOSITION Ponsus Pharma AB (SE) 2004-10-06 EP disclosed
WO-2003055454-A1 NEW COMPOSITION PONSUS PHARMA AB (SE) 2003-07-10 WO disclosed