SCHEMBL6832341

SCHEMBL6832341

COc1cnc(Cl)c(Nc2c(C#N)cnc3cc(OCCCN4CCOCC4)c(OC)cc23)n1

nearest known ligand 0.72

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SRC P12931 12/20 0.72
ABL1 P00519 2/20 0.72
BCR P11274 2/20 0.72
MAP2K1 Q02750 7/20 0.70
FYN P06241 1/20 0.70
EGFR P00533 1/20 0.69
ERBB2 P04626 1/20 0.69
RAF1 P04049 1/20 0.65
MAPK3 P27361 1/20 0.65
MAPK1 P28482 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6684408 0.91 SRC (0.76) SRCABL1BCRMAP2K1FYN
SCHEMBL6832310 0.86 SRC (0.74) SRCABL1BCRMAP2K1FYN
SCHEMBL6834093 0.86 SRC (0.57) SRCABL1BCREGFRERBB2
SCHEMBL6685924 0.85 SRC (0.83) SRCABL1BCRMAP2K1FYN
SCHEMBL6930676 0.84 SRC (0.57) SRCABL1BCREGFRERBB2
SCHEMBL5201099 0.82 SRC (1.00) SRCABL1BCRMAP2K1FYN
SCHEMBL4485027 0.82 SRC (0.71) SRCABL1BCRMAP2K1FYN
SCHEMBL6383141 0.81 EGFR (1.00) SRCABL1BCRMAP2K1FYN
SCHEMBL6382257 0.81 SRC (0.76) SRCABL1BCRMAP2K1FYN
SCHEMBL6381057 0.81 SRC (0.76) SRCABL1BCRMAP2K1FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004108703-A1 PYRAZINYL 3-CYANOQUINOLINE DERIVATIVES FOR USE IN THE TREATMENT OF TUMOURS ASTRAZENECA AB (SE) 2004-12-16 WO disclosed