SCHEMBL6833719

SCHEMBL6833719

COc1cc(NC(=S)NC2CCC(Nc3nc4c(c(N(C)C)n3)CCCC4)CC2)cc(OC)c1OC

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.38
TP53 P04637 1/20 0.38
ADRA2A P08913 1/20 0.37
MCHR1 Q99705 1/20 0.37
ALDH1A1 P00352 4/20 0.37
HTT P42858 1/20 0.37
KDM4E B2RXH2 3/20 0.37
POLB P06746 1/20 0.37
RAB9A P51151 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GAA P10253 1/20 0.36
NPC1 O15118 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6457954 1.00 MAPT (0.38) MAPTTP53ADRA2AMCHR1ALDH1A1
SCHEMBL6460993 0.90 SMN1; SMN2 (0.40) MAPTTP53ADRA2AMCHR1ALDH1A1
SCHEMBL6460982 0.90 SMN1; SMN2 (0.40) MAPTTP53ADRA2AMCHR1ALDH1A1
SCHEMBL6456641 0.89 TP53 (0.41) MAPTTP53ADRA2AMCHR1ALDH1A1
SCHEMBL6456647 0.89 TP53 (0.41) MAPTTP53ADRA2AMCHR1ALDH1A1
SCHEMBL6872800 0.89 MCHR1 (0.46) MAPTADRA2AMCHR1POLBRAB9A
SCHEMBL6872807 0.89 MCHR1 (0.46) MAPTADRA2AMCHR1POLBRAB9A
SCHEMBL6875342 0.86 GAA (0.42) MAPTADRA2AMCHR1ALDH1A1POLB
SCHEMBL6875336 0.86 GAA (0.42) MAPTADRA2AMCHR1ALDH1A1POLB
SCHEMBL6868226 0.85 BCHE (0.46) MAPTTP53ADRA2AMCHR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087669-A1 NOVEL QUINOLINE, TETRAHYDROQUINAZOLINE, AND PYRIMIDINE DERIVATIVES AND METHODS OF TREATMENT RELATED TO THE USE THEREOF TAISHO PHARMACEUTICAL CO. LTD. (JP) 2004-10-14 WO claimed
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP claimed
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed