SCHEMBL6834302

SCHEMBL6834302

O=C(N[C@H]1CCCC[C@H]1C(=O)O)c1cc2ccc(Br)cc2[nH]1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.56
F10 P00742 2/20 0.45
MLLT1 Q03111 1/20 0.44
HRH4 Q9H3N8 1/20 0.44
CCKBR P32239 2/20 0.42
CGAS Q8N884 1/20 0.41
GRK2 P25098 1/20 0.40
CASP6 P55212 1/20 0.40
CASP8 Q14790 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PYGL P06737 1/20 0.39
PYGM P11217 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6832859 0.91 MLLT1 (0.52) DRD4F10MLLT1HRH4CCKBR
SCHEMBL15506751 0.86 DRD4 (0.65) DRD4F10HRH4
SCHEMBL5260262 0.86 F10 (0.59) F10PYGLPYGM
SCHEMBL5256019 0.84 CCKBR (0.57) MLLT1CCKBRCGASPYGLPYGM
SCHEMBL27558367 0.84 CCKBR (0.57) MLLT1CCKBRCGASPYGLPYGM
SCHEMBL29176327 0.84 MLLT1 (0.61) DRD4MLLT1HRH4
SCHEMBL6839437 0.83 DRD4 (0.50) DRD4F10MLLT1HRH4PYGL
SCHEMBL5256902 0.83 F10 (0.43) DRD4F10MLLT1CCKBRCGAS
SCHEMBL5255542 0.83 KMT2A (0.55) HRH4
SCHEMBL29176357 0.83 MLLT1 (0.60) DRD4MLLT1HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6759428-B2 SUCH AS N-((1,2)-2-(((CYANO(CYCLOPROPYL)METHYL)AMINO)CARBONYL) CYCLOHEXYL)-1H-INDOLE-2-CARBOXAMIDE; CATHEPSIN K INHIBITORS ROCHE PALO ALTO LLC 2004-07-06 US disclosed