SCHEMBL6836229

SCHEMBL6836229

CC(=O)O[C@@]1(C(=O)CO)CC[C@H]2[C@@H]3C[C@H](C)C4=CC(=O)C=C[C@]4(C)[C@H]3[C@@H](O)C[C@@]21C

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.73
PGR P06401 7/20 0.73
NR3C1 P04150 7/20 0.73
HIF1A Q16665 5/20 0.73
HSD17B10 Q99714 4/20 0.73
ABCB11 O95342 4/20 0.73
ALDH1A1 P00352 1/20 0.73
ABCC4 O15439 1/20 0.73
NR1I2 O75469 1/20 0.73
PDE4D Q08499 1/20 0.73
AR P10275 3/20 0.68
F2 P00734 1/20 0.68
CYP2C19 P33261 2/20 0.51
NR3C2 P08235 2/20 0.51
TNF P01375 1/20 0.51
IL6 P05231 1/20 0.51
SERPINA6 P08185 1/20 0.51
GLUL P15104 1/20 0.51
ADAM17 P78536 1/20 0.51
GPBAR1 Q8TDU6 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1371249 1.00 CYP3A4 (0.73) CYP3A4PGRNR3C1HIF1AHSD17B10
SCHEMBL11878275 1.00 CYP3A4 (0.73) CYP3A4PGRNR3C1HIF1AHSD17B10
SCHEMBL11878266 1.00 CYP3A4 (0.73) CYP3A4PGRNR3C1HIF1AHSD17B10
SCHEMBL6836230 1.00 CYP3A4 (0.73) CYP3A4PGRNR3C1HIF1AHSD17B10
SCHEMBL6856646 0.92 PGR (0.71) CYP3A4PGRNR3C1HIF1AHSD17B10
SCHEMBL10904456 0.92 PGR (0.71) CYP3A4PGRNR3C1HIF1AHSD17B10
SCHEMBL6856651 0.92 PGR (0.71) CYP3A4PGRNR3C1HIF1AHSD17B10
SCHEMBL10527423 0.92 PGR (0.71) CYP3A4PGRNR3C1HIF1AHSD17B10
SCHEMBL11126257 0.92 PGR (0.79) CYP3A4PGRNR3C1HIF1AHSD17B10
SCHEMBL10906704 0.92 PGR (0.79) CYP3A4PGRNR3C1HIF1AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6828120-B2 Preparation of 11 beta ,17 alpha ,21- trihydroxy-6 alpha -methylpregna-1,4-diene-3,20-dione 21-acetate; obtain chemical intermediates, incubate reaction mix and enzymes, recover product PHARMACIA AND UPJOHN COMPANY 2004-12-07 US disclosed
US-20040006240-A1 Process to prepare 11beta,17alpha ,21-trihydroxy-6alpha-methylpregna-1,4-diene-3,20-dione 21-acetate PHARMACIA & UPJOHN COMPANY 2004-01-08 US disclosed
US-20030044885-A1 Process to prepare 11beta, 17alpha,21-trihydroxy-6alpha-methylpregna-1,4-diene-3,20-dione 21-acetate CRIA, INC. 2003-03-06 US disclosed
US-20030013900-A1 Process to prepare11beta,17alpha, 21-trihydroxy-6alpha-methylpregna-1,4-diene-3,20-dione 21-acetate PHARMACIA & UPJOHN COMPANY 2003-01-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030013900-A1 Process to prepare11beta,17alpha, 21-trihydroxy-6alpha-methylpregna-1,4-diene-3,20-dione 21-acetate CYP17A1, CYP51A1, CYP4A11 CYP3A4 102/4885PGR 447/4885NR3C1 118/4885
US-20030044885-A1 Process to prepare 11beta, 17alpha,21-trihydroxy-6alpha-methylpregna-1,4-diene-3,20-dione 21-acetate CYP17A1, CYP51A1, HSD17B11 CYP3A4 86/4885PGR 339/4885NR3C1 103/4885
US-20040006240-A1 Process to prepare 11beta,17alpha ,21-trihydroxy-6alpha-methylpregna-1,4-diene-3,20-dione 21-acetate CYP17A1, CYP51A1, HSD17B11 CYP3A4 96/4885PGR 448/4885NR3C1 117/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.