SCHEMBL6836698

SCHEMBL6836698

Cc1nc(C(=O)[N+]2(C)CCNC(CNC(=O)c3cccc4occc34)C2)c(-c2ccc(F)cc2)s1

nearest known ligand 0.60

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 20/20 0.60
HCRTR2 O43614 17/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7068626 0.89 HCRTR1 (0.49) HCRTR1HCRTR2
SCHEMBL7068936 0.86 HCRTR1 (0.45) HCRTR1HCRTR2
SCHEMBL4829047 0.85 HCRTR1 (0.43) HCRTR1HCRTR2
SCHEMBL7132041 0.85 HCRTR1 (0.43) HCRTR1HCRTR2
SCHEMBL5802846 0.83 HCRTR1 (0.64) HCRTR1HCRTR2
SCHEMBL6835547 0.81 HCRTR1 (0.40) HCRTR1HCRTR2
SCHEMBL1398707 0.77 HCRTR1 (0.90) HCRTR1HCRTR2
SCHEMBL1398620 0.77 HCRTR1 (0.90) HCRTR1HCRTR2
SCHEMBL1398677 0.77 HCRTR1 (0.90) HCRTR1HCRTR2
SCHEMBL6832457 0.77 HCRTR1 (0.43) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441729-A1 PIPERAZINE BIS-AMIDE DERIVATIVES AND THEIR USE AS ANTAGONISTS OF THE OREXIN RECEPTOR SMITHKLINE BEECHAM PLC (GB) 2004-08-04 EP disclosed
WO-2003041711-A1 PIPERAZINE BIS-AMIDE DERIVATIVES AND THEIR USE AS ANTAGONISTS OF THE OREXIN RECEPTOR SMITHKLINE BEECHAM P.L.C. (GB) 2003-05-22 WO disclosed