SCHEMBL6837299

SCHEMBL6837299

CC(O)c1sc(NC(=O)OC(C)(C)C)nc1Br

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
LCK P06239 14/20 0.46
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
PI4KB Q9UBF8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27459853 0.89 LCK (0.44) LCKCA1CA2PI4KB
SCHEMBL34467451 0.80 LCK (0.43) LCKPI4KB
SCHEMBL1563222 0.78 LCK (0.48) LCKCA1CA2PI4KB
SCHEMBL15186149 0.77 LCK (0.53) LCKCA1CA2PI4KB
SCHEMBL12056453 0.77 LCK (0.53) LCKCA1CA2PI4KB
SCHEMBL21394961 0.76 LCK (0.42) LCK
SCHEMBL29357021 0.76 LCK (0.42) LCK
SCHEMBL31488298 0.76 LCK (0.52) LCKCA1CA2PI4KB
SCHEMBL367235 0.76 CA1 (0.47) LCKCA1CA2PI4KB
SCHEMBL24736315 0.75 LCK (0.50) LCKCA1CA2PI4KB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025151517-A1 THIAZOLE COMPOUNDS, COMPOSITIONS AND METHODS OF TREATING DISORDERS ASSOCIATED WITH MISSFOLDING OF ALPHA-SYNUCLEIN PROTEIN WAVEBREAK THERAPEUTICS LIMITED (US) 2025-07-17 WO disclosed
US-20130210807-A1 Tricyclic Compounds as Allosteric Modulators of Metabotropic Glutamate Receptors. MERCK SHARP & DOHME CORP. 2013-08-15 US disclosed
WO-2012006760-A1 TRICYCLIC COMPOUNDS AS ALLOSTERIC MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS MERCK SHARP & DOHME CORP. (US) 2012-01-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130210807-A1 Tricyclic Compounds as Allosteric Modulators of Metabotropic Glutamate Receptors. GRM3, GRM6, GRM1 LCK 2208/4885CA1 1272/4885CA2 996/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.