SCHEMBL6844115

SCHEMBL6844115

NC(=O)CCc1ccc2[nH]ccc2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.55
HDAC8 Q9BY41 2/20 0.55
CAPN1 P07384 1/20 0.47
CTNNB1 P35222 4/20 0.47
WNT3A P56704 4/20 0.47
F2 P00734 1/20 0.46
USP2 O75604 1/20 0.44
GAA P10253 1/20 0.44
ALOX15 P16050 1/20 0.44
RAD51 Q06609 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
MAOB P27338 1/20 0.42
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21274689 0.87 BACE1 (0.50) HDAC1HDAC8CAPN1HDAC3HDAC4
SCHEMBL6263512 0.85 HDAC1 (0.56) HDAC1HDAC8CTNNB1WNT3A
SCHEMBL4883079 0.84 HDAC1 (0.55) HDAC1HDAC8CTNNB1WNT3AUSP2
SCHEMBL9225433 0.83 HDAC1 (0.54) HDAC1HDAC8CTNNB1WNT3AF2
SCHEMBL30006673 0.83 HDAC1 (0.54) HDAC1HDAC8CTNNB1WNT3AF2
SCHEMBL14820597 0.82 HDAC1 (0.71) HDAC1HDAC8CTNNB1WNT3AF2
SCHEMBL8666600 0.80 HDAC1 (0.55) HDAC1HDAC8CTNNB1WNT3AF2
SCHEMBL6303056 0.80 HDAC1 (0.51) HDAC1HDAC8CTNNB1WNT3AUSP2
SCHEMBL15901671 0.80 HDAC1 (0.54) HDAC1HDAC8CTNNB1WNT3AMAOB
SCHEMBL28325361 0.79 HDAC1 (0.60) HDAC1HDAC8CTNNB1WNT3AUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115279782-A Peptide inhibitors of interleukin-23 receptor and their use for the treatment of inflammatory diseases 詹森生物科技公司 2022-11-01 CN disclosed
EP-1330457-B1 CYCLOPENTA[B][1,4] DIAZEPINO[6,7,1-HI]INDOLES AS 5HT2C ANTAGONISTS WYETH CORP (US) 2004-10-20 EP disclosed
EP-0997474-A1 Antithrombotic agents PFIZER INC. (US) 2000-05-03 EP disclosed
CN-1208413-A Gonadotropin releasing hormone antagonists MERCK & CO INC (US) 1999-02-17 CN disclosed