SCHEMBL6844490

SCHEMBL6844490

CC(N)/C=N/C(=O)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
LMNA P02545 1/20 0.39
XBP1 P17861 1/20 0.39
ATM Q13315 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TSHR P16473 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
CYP2C19 P33261 2/20 0.39
POLB P06746 1/20 0.39
CYP3A4 P08684 1/20 0.39
PARP1 P09874 1/20 0.39
RECQL P46063 1/20 0.39
BLM P54132 1/20 0.39
PMP22 Q01453 1/20 0.39
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TAAR1 Q96RJ0 1/20 0.38
ALDH1A1 P00352 4/20 0.37
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8051024 0.85 MAPT (0.41) MAPTSMN1; SMN2LMNAXBP1ATM
SCHEMBL4516672 0.75 TSHR (0.43) MAPTSMN1; SMN2LMNAXBP1ATM
SCHEMBL15689787 0.74 TDP1 (0.46) MAPTSMN1; SMN2LMNATSHRTDP1
SCHEMBL13341652 0.74 CES1 (0.44) MAPTSMN1; SMN2TSHRTDP1CYP2C19
SCHEMBL4900468 0.74 TDP1 (0.46) MAPTSMN1; SMN2LMNATSHRTDP1
SCHEMBL28825945 0.74 CES1 (0.44) MAPTSMN1; SMN2TSHRTDP1CYP2C19
SCHEMBL4560875 0.71 CES1 (0.45) MAPTSMN1; SMN2LMNAATMNPSR1
SCHEMBL791662 0.70 CES1 (0.44) MAPTSMN1; SMN2LMNAATMTSHR
SCHEMBL6384300 0.70 MAPT (0.45) MAPTSMN1; SMN2LMNAXBP1ATM
SCHEMBL791663 0.70 CES1 (0.44) MAPTSMN1; SMN2LMNAATMTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079114-A1 PTERIDINONES AS INHIBITORS OF POLO - LIKE KINASE ELAN PHARMACEUTICALS, INC. (US) 2011-06-30 WO disclosed
WO-2011079118-A1 PTERIDINONES AS INHIBITORS OF POLO-LIKE KINASE ELAN PHARMACEUTICALS, INC (US) 2011-06-30 WO disclosed