SCHEMBL8051024

SCHEMBL8051024

CC(C)/C=N\C(=O)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 1/20 0.41
XBP1 P17861 1/20 0.41
ATM Q13315 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
ALDH1A1 P00352 5/20 0.39
CES2 O00748 3/20 0.39
CES1 P23141 3/20 0.39
TSHR P16473 3/20 0.39
DAO P14920 1/20 0.39
NAPRT Q6XQN6 1/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
RAB9A P51151 1/20 0.39
TDP1 Q9NUW8 3/20 0.39
MAPK1 P28482 1/20 0.39
GAA P10253 1/20 0.38
PGR P06401 1/20 0.38
ADRA2A P08913 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6844490 0.85 MAPT (0.39) MAPTSMN1; SMN2LMNAXBP1ATM
SCHEMBL28402297 0.79 ALDH1A1 (0.49) MAPTSMN1; SMN2LMNAALDH1A1NPC1
SCHEMBL13341652 0.77 CES1 (0.44) MAPTSMN1; SMN2ALDH1A1CES2CES1
SCHEMBL28825945 0.77 CES1 (0.44) MAPTSMN1; SMN2ALDH1A1CES2CES1
SCHEMBL4560875 0.73 CES1 (0.45) MAPTSMN1; SMN2LMNAATMNPSR1
SCHEMBL791663 0.72 CES1 (0.44) MAPTSMN1; SMN2LMNAATMALDH1A1
SCHEMBL4900468 0.72 TDP1 (0.46) MAPTSMN1; SMN2LMNAALDH1A1CES2
SCHEMBL791662 0.72 CES1 (0.44) MAPTSMN1; SMN2LMNAATMALDH1A1
SCHEMBL15689787 0.72 TDP1 (0.46) MAPTSMN1; SMN2LMNAALDH1A1CES2
SCHEMBL6384300 0.72 MAPT (0.45) MAPTSMN1; SMN2LMNAXBP1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009075778-A2 NONPEPTIDIC INHIBITORS OF CRUZAIN THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2009-06-18 WO disclosed