SCHEMBL6844769

SCHEMBL6844769

O=C(O)Cc1nn(-c2ccccc2F)cc1-c1ccc(Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.46
DRD2 P14416 1/20 0.46
PTGS1 P23219 2/20 0.42
PTGS2 P35354 2/20 0.42
FABP4 P15090 1/20 0.42
PTGES O14684 2/20 0.42
ALOX5 P09917 1/20 0.42
RAB9A P51151 2/20 0.40
CNR1 P21554 2/20 0.40
SUCNR1 Q9BXA5 1/20 0.39
NOTUM Q6P988 1/20 0.39
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38
PTGDR2 Q9Y5Y4 3/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
HPGD P15428 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11761156 0.91 PTGS1 (0.47) KDM4EPTGS1PTGS2FABP4RAB9A
SCHEMBL11469421 0.84 MAPT (0.43) PTGS1PTGS2RAB9AALDH1A1SMN1; SMN2
SCHEMBL11408123 0.84 KDM4E (0.64) KDM4EDRD2PTGS2PTGESALOX5
SCHEMBL11763324 0.81 BCHE (0.43) KDM4EDRD2FABP4RAB9ANOTUM
SCHEMBL11762851 0.81 KDM4E (0.57) KDM4EDRD2PTGS2PTGESALOX5
SCHEMBL11443525 0.81 KDM4E (0.56) KDM4EDRD2PTGS2PTGESALOX5
Pirazolac SCHEMBL153631 0.81 KDM4E (0.51) KDM4EDRD2PTGS2PTGESALOX5
Pirazolac SCHEMBL10952997 0.80 KDM4E (0.50) KDM4EDRD2PTGS2PTGESALOX5
SCHEMBL11766518 0.78 RAB9A (0.51) RAB9ANOTUMSMN1; SMN2NPC1MAPT
SCHEMBL11767431 0.78 KDM4E (0.43) KDM4EDRD2PTGESALOX5RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0022906-A1 Process for the preparation of pyrazole derivatives SCHERING AKTIENGESELLSCHAFT (DE) 1981-01-28 EP claimed
US-20040242597-A1 Combination NYCOMED GMBH (DE) 2004-12-02 US disclosed
EP-0022906-B1 PROCESS FOR THE PREPARATION OF PYRAZOLE DERIVATIVES SCHERING AKTIENGESELLSCHAFT (DE) 1984-08-08 EP disclosed
EP-0022906-A1 Process for the preparation of pyrazole derivatives SCHERING AKTIENGESELLSCHAFT (DE) 1981-01-28 EP disclosed