SCHEMBL6845259

SCHEMBL6845259

CCCN1CCN(c2nc(-c3ccnc(NO)c3)cnc2N)CC1

nearest known ligand 0.59

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 10/20 0.59
ROCK1 Q13464 9/20 0.59
NEK2 P51955 7/20 0.41
PTPN11 Q06124 1/20 0.40
ACHE P22303 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2322669 0.73 ROCK2 (0.72) ROCK2ROCK1NEK2
SCHEMBL2321088 0.73 ROCK2 (0.87) ROCK2ROCK1NEK2
SCHEMBL12439974 0.70 ROCK2 (1.00) ROCK2ROCK1NEK2
Hydrochloric Acid SCHEMBL2320003 0.70 ROCK2 (0.98) ROCK2ROCK1NEK2
SCHEMBL2325042 0.69 ROCK2 (0.75) ROCK2ROCK1NEK2
SCHEMBL2321462 0.69 ROCK2 (0.71) ROCK2ROCK1NEK2
SCHEMBL988824 0.67 ROCK2 (0.69) ROCK2ROCK1
SCHEMBL3513029 0.66 ROCK2 (1.00) ROCK2ROCK1
SCHEMBL2323120 0.66 ROCK2 (0.65) ROCK2ROCK1NEK2
SCHEMBL2321276 0.65 ROCK2 (0.67) ROCK2ROCK1NEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7867999-B1 Hydroxyamino- and amino-substituted pyridine analogs for treating rho kinase-mediated diseases and conditions ALCON RESEARCH, LTD. (US) 2011-01-11 US disclosed