SCHEMBL6845267

SCHEMBL6845267

CNC(C)c1ccc(C(=O)Nc2ccncc2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.71
ROCK1 Q13464 2/20 0.71
KDM4E B2RXH2 1/20 0.67
L3MBTL1 Q9Y468 1/20 0.67
KMT2A Q03164 3/20 0.58
NT5E P21589 1/20 0.58
GAA P10253 1/20 0.57
JAK2 O60674 1/20 0.57
TYK2 P29597 1/20 0.57
POLB P06746 2/20 0.55
STAT3 P40763 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
LMNA P02545 3/20 0.55
ALDH1A1 P00352 2/20 0.55
MAPK1 P28482 2/20 0.55
TP53 P04637 1/20 0.55
HTT P42858 1/20 0.53
MAPT P10636 1/20 0.52
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30192651 0.86 ROCK2 (0.77) ROCK2ROCK1KDM4EL3MBTL1KMT2A
SCHEMBL5460526 0.84 ROCK2 (0.75) ROCK2ROCK1KDM4EL3MBTL1KMT2A
SCHEMBL1554113 0.83 ROCK2 (1.00) ROCK2ROCK1KDM4EL3MBTL1KMT2A
SCHEMBL1553349 0.83 ROCK2 (1.00) ROCK2ROCK1KDM4EL3MBTL1KMT2A
SCHEMBL1553353 0.83 ROCK2 (1.00) ROCK2ROCK1KDM4EL3MBTL1KMT2A
SCHEMBL6558035 0.82 ROCK2 (0.67) ROCK2ROCK1KDM4EL3MBTL1KMT2A
SCHEMBL6558041 0.82 ROCK2 (0.67) ROCK2ROCK1KDM4EL3MBTL1KMT2A
Hydrochloric Acid SCHEMBL1770829 0.82 ROCK2 (1.00) ROCK2ROCK1KDM4EL3MBTL1KMT2A
Hydrochloric Acid SCHEMBL2474313 0.82 ROCK2 (1.00) ROCK2ROCK1KDM4EL3MBTL1KMT2A
Hydrochloric Acid SCHEMBL1770831 0.82 ROCK2 (1.00) ROCK2ROCK1KDM4EL3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7867999-B1 Hydroxyamino- and amino-substituted pyridine analogs for treating rho kinase-mediated diseases and conditions ALCON RESEARCH, LTD. (US) 2011-01-11 US disclosed