SCHEMBL6846633

SCHEMBL6846633

COc1ccc(OC)c2ncc(CO)cc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.47
POLB P06746 1/20 0.47
RAB9A P51151 1/20 0.47
PDE4A P27815 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
FYN P06241 2/20 0.42
SYK P43405 1/20 0.39
IRAK4 Q9NWZ3 1/20 0.39
PDE1B Q01064 1/20 0.39
ATP4A P20648 1/20 0.39
ATP4B P51164 1/20 0.39
HPGDS O60760 1/20 0.38
DPP4 P27487 1/20 0.37
TOP2A P11388 2/20 0.36
TOP2B Q02880 2/20 0.36
HSD17B10 Q99714 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13313452 0.81 SYK (0.43) NPC1POLBRAB9AFYNSYK
SCHEMBL11971452 0.78 PDE10A (0.53) NPC1POLBRAB9AFYNTOP2A
SCHEMBL28128228 0.77 CA2 (0.41) RAB9APDE4APDE4BPDE4CPDE4D
SCHEMBL27505904 0.75 PDE4A (0.39) NPC1PDE4APDE4BPDE4CPDE4D
SCHEMBL4700757 0.73 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DATP4A
SCHEMBL7822137 0.72 CA12 (0.50) RAB9AHPGDS
SCHEMBL4698817 0.72 PDE4A (0.64) PDE4APDE4BPDE4CPDE4D
SCHEMBL9360729 0.72 MEN1 (0.49) NPC1POLBRAB9APDE4APDE4B
SCHEMBL19330511 0.72 NPC1 (0.48) NPC1POLBRAB9APDE4APDE4B
SCHEMBL21499282 0.72 NPC1 (0.48) NPC1POLBRAB9APDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1202992-B1 ASCIDIDEMIN DERIVATIVES AND THEIR THERAPEUTIC APPLICATIONS CEPHALON FRANCE (FR) 2004-09-15 EP disclosed
EP-1202992-A2 ASCIDIDEMIN DERIVATIVES AND THEIR THERAPEUTIC APPLICATIONS LABORATOIRE L. LAFON (FR) 2002-05-08 EP disclosed
WO-2001012631-A2 ASCIDIDEMIN DERIVATIVES AND THEIR THERAPEUTIC APPLICATIONS LABORATOIRE L. LAFON (FR) 2001-02-22 WO disclosed