SCHEMBL6846771

SCHEMBL6846771

CCCOc1ccc(-c2[nH]c3nccnc3c2CCC(=O)O)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 17/20 0.61
GSK3B P49841 17/20 0.61
CDK1 P06493 16/20 0.61
CCNB2 O95067 15/20 0.61
CCNB1 P14635 15/20 0.61
CCNB3 Q8WWL7 15/20 0.61
CDK5 Q00535 11/20 0.61
CDK5R1 Q15078 10/20 0.61
CDK2 P24941 3/20 0.58
CCNE1 P24864 2/20 0.58
ZAP70 P43403 1/20 0.58
PTK2B Q14289 1/20 0.58
MAPK8 P45983 3/20 0.55
CCNE2 O96020 1/20 0.55
INSR P06213 1/20 0.55
CFTR P13569 1/20 0.55
CCNA2 P20248 1/20 0.55
MAPK3 P27361 1/20 0.55
MAPK1 P28482 1/20 0.55
MAPK9 P45984 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6851003 0.91 CDK5 (0.61) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL6852671 0.89 GSK3A (0.58) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL1777822 0.87 GSK3A (0.72) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL1777025 0.84 GSK3A (0.55) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL6852911 0.84 GSK3A (0.67) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL1778366 0.82 GSK3A (0.70) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL1777830 0.81 GSK3A (0.59) GSK3AGSK3BCDK1CCNB2CCNB1
Iodide SCHEMBL6852377 0.78 GSK3A (0.58) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL1777268 0.76 GSK3A (0.69) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL1777706 0.76 GSK3A (0.55) GSK3AGSK3BCDK1CCNB2CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397360-A1 AZAINDOLES Aventis Pharma Limited (GB) 2004-03-17 EP disclosed
WO-2003000688-A1 AZAINDOLES AVENTIS PHARMA LIMITED (GB) 2003-01-03 WO disclosed
EP-1263759-A2 AZAINDOLES Aventis Pharma Limited (GB) 2002-12-11 EP disclosed
WO-2001047922-A2 AZAINDOLES AVENTIS PHARMA LIMITED (GB) 2001-07-05 WO disclosed