SCHEMBL6852208

SCHEMBL6852208

O=C(O)N1CCc2c(n3c4c(cc(F)c(F)c24)OCC3)CC1

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
MCL1 Q07820 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7674690 0.90 PTGDR (0.31) PTGDR2
SCHEMBL7673244 0.88 MAPT (0.30) HTR2AHTR2C
SCHEMBL7676778 0.85 HTR2C (0.37) HTR2AHTR2CPTGDR2MCL1
SCHEMBL6851580 0.82 MCL1 (0.32) HTR2AHTR2CMCL1
SCHEMBL6853636 0.81 PTGDR2 (0.49) PTGDR2
SCHEMBL7673579 0.81 HTR2A (0.38) HTR2AHTR2CPTGDR2MCL1
Maleic Acid SCHEMBL6482229 0.78 HTR2C (0.45) HTR2AHTR2C
SCHEMBL7679724 0.78 HTR2A (0.36) HTR2AHTR2CPTGDR2MCL1
SCHEMBL6497051 0.78 HTR2A (0.34) HTR2AHTR2CMCL1
SCHEMBL6847402 0.77 HTR2C (0.53) HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1173440-B1 TETRACYCLIC AZEPINOINDOLE COMPOUNDS AS 5-HT RECEPTOR LIGANDS UPJOHN CO (US) 2004-09-15 EP claimed