SCHEMBL6852593

SCHEMBL6852593

OCC(F)=Cc1cnc(-c2ccccc2)nc1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.47
NFKB1 P19838 2/20 0.47
RAB9A P51151 2/20 0.47
NFKB2 Q00653 2/20 0.47
RELA Q04206 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
HPGDS O60760 15/20 0.40
CYP11B1 P15538 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6852587 1.00 NPC1 (0.47) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL6852590 1.00 NPC1 (0.47) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL6852121 0.81 NPC1 (0.48) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL6852124 0.81 NPC1 (0.48) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL6854217 0.80 HDAC4 (0.35) NPC1RAB9ASMN1; SMN2
SCHEMBL6881060 0.80 HDAC4 (0.35) NPC1RAB9ASMN1; SMN2
SCHEMBL6881056 0.80 HDAC4 (0.35) NPC1RAB9ASMN1; SMN2
SCHEMBL6879073 0.79 ADRB2 (0.42) NPC1RAB9A
SCHEMBL6276439 0.79 ADRB2 (0.42) NPC1RAB9A
SCHEMBL6309957 0.79 ADRB2 (0.42) NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825170-B2 ERYTHROMYCIN TYPE MACROLIDE WITH A FUSED OXAZOLONE RING ORTHO-MCNEIL PHARMACEUTICAL, INC. 2004-11-30 US disclosed
EP-1453847-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS Ortho-Mcneil Pharmaceutical, Inc. (US) 2004-09-08 EP disclosed
WO-2003050132-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2003-06-19 WO disclosed