SCHEMBL6852901

SCHEMBL6852901

OC/C=C/c1csc(-c2ncccn2)c1

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
CYP3A4 P08684 1/20 0.35
RECQL P46063 1/20 0.35
RHOA P61586 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6852906 1.00 ALDH1A1 (0.35) ALDH1A1CYP3A4RECQLRHOAIRAK4
SCHEMBL6853980 0.83 KDM4E (0.43) ALDH1A1CYP3A4RECQLRHOA
SCHEMBL6853984 0.83 KDM4E (0.43) ALDH1A1CYP3A4RECQLRHOA
SCHEMBL6851976 0.78 CYP19A1 (0.32)
SCHEMBL6852127 0.76 PIM2 (0.34) ALDH1A1CYP3A4RECQL
SCHEMBL6852115 0.76 PIM2 (0.34) ALDH1A1CYP3A4RECQL
SCHEMBL6876939 0.75 ALDH1A1 (0.37) ALDH1A1
SCHEMBL6876943 0.75 ALDH1A1 (0.37) ALDH1A1
SCHEMBL6851987 0.75
SCHEMBL6851982 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825170-B2 ERYTHROMYCIN TYPE MACROLIDE WITH A FUSED OXAZOLONE RING ORTHO-MCNEIL PHARMACEUTICAL, INC. 2004-11-30 US disclosed
EP-1463804-A1 IMPROVED GAMETE RECRUITMENT AND DEVELOPMENTAL COMPETENCE IN MAMMALS BY INHIBITING THE DE NOVO STEROL BIOSYNTHESIS AND/OR PROMOTING STEROL EFFLUX Rigshospitalet (DK) 2004-10-06 EP disclosed
EP-1453847-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS Ortho-Mcneil Pharmaceutical, Inc. (US) 2004-09-08 EP disclosed
WO-2003055991-A1 IGAMETE RECRUITMENT AND DEVELOPMENTAL COMPETENCE IN MAMMALS BY INHIBITING THE DE NOVO STEROL BIOSYNTHESIS AND/OR PROMOTING STEROL EFFLUX RIGSHOSPITALET (DK) 2003-07-10 WO disclosed
WO-2003050132-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2003-06-19 WO disclosed