SCHEMBL6853307

SCHEMBL6853307

CN(C)CC(=O)N1CCN(Cc2c(-c3ccccc3)nc3ccccc3c2C(=O)O)CC1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 17/20 0.54
TACR2 P21452 10/20 0.54
KCNH2 Q12809 7/20 0.52
OPRM1 P35372 5/20 0.50
TSHR P16473 1/20 0.47
PDE10A Q9Y233 1/20 0.47
LMNA P02545 1/20 0.47
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6851699 0.86 TACR3 (0.67) TACR3TACR2KCNH2OPRM1TSHR
SCHEMBL5461424 0.85 TACR2 (0.53) TACR3TACR2KCNH2OPRM1PDE10A
SCHEMBL6853049 0.84 TACR3 (0.58) TACR3TACR2KCNH2OPRM1TSHR
SCHEMBL6853022 0.84 TACR3 (0.51) TACR3TACR2KCNH2OPRM1
SCHEMBL6855404 0.84 TACR2 (0.54) TACR3TACR2KCNH2OPRM1PDE10A
SCHEMBL6848956 0.83 TACR2 (0.61) TACR3TACR2KCNH2OPRM1TSHR
SCHEMBL6851678 0.83 TACR3 (0.69) TACR3TACR2KCNH2OPRM1
SCHEMBL27583479 0.83 TACR2 (0.53) TACR3TACR2KCNH2OPRM1TSHR
SCHEMBL6853618 0.83 TACR2 (0.55) TACR3TACR2KCNH2OPRM1TSHR
SCHEMBL5429087 0.82 TACR2 (0.56) TACR3TACR2KCNH2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6780875-B2 RESPIRATORY SYSTEM DISORDERS; ANTIINFLAMMATORY AGENTS; PSYCHOLOGICAL DISORDERS SMITHKLINE BEECHAM S.P.A. (IT) 2004-08-24 US claimed
US-6780875-B2 RESPIRATORY SYSTEM DISORDERS; ANTIINFLAMMATORY AGENTS; PSYCHOLOGICAL DISORDERS SMITHKLINE BEECHAM S.P.A. (IT) 2004-08-24 US disclosed