SCHEMBL6853497

SCHEMBL6853497

CC1(c2ccc(O)cc2)NC(=O)Nc2ccc(I)cc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.40
MMP9 P14780 1/20 0.40
CHRM2 P08172 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
KCNH2 Q12809 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
AKR1B1 P15121 1/20 0.36
KDM4E B2RXH2 1/20 0.35
GAA P10253 1/20 0.35
GFER P55789 1/20 0.35
HTR6 P50406 2/20 0.33
TGM2 P21980 1/20 0.33
CES1 P23141 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6853483 0.83 PDE7A (0.48) MMP2MMP9CHRM2ADORA3KCNH2
SCHEMBL8471852 0.83 PDE7A (0.48) MMP2MMP9CHRM2ADORA3KCNH2
SCHEMBL1408090 0.83 PDE7A (0.48) MMP2MMP9CHRM2ADORA3KCNH2
SCHEMBL5483163 0.74 CHRM2 (0.62) MMP2MMP9CHRM2ADORA3KCNH2
SCHEMBL21939542 0.70 AKR1B1 (0.46) MMP2MMP9KCNH2CA12CA1
SCHEMBL19605042 0.70 AKR1B1 (0.46) MMP2MMP9KCNH2CA12CA1
SCHEMBL10131744 0.69 LMNA (0.51) MMP2MMP9KCNH2AKR1B1HTR6
SCHEMBL10116540 0.69 PDK2 (0.55)
SCHEMBL31238681 0.69 PDK2 (0.55)
SCHEMBL21940203 0.69 PDE7A (0.50) AKR1B1GAAHTR6PDE7A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745785-B1 Pharmaceutical composition for preventing or treating cerebral oedema BIOCODEX (FR) 2011-03-09 EP disclosed