SCHEMBL6856819

SCHEMBL6856819

CC(C)NC(=O)Cc1cc2cc(OC3CCNCC3)ccc2nc1-c1ccc(F)c(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AVPR1B P47901 4/20 0.41
CHRM1 P11229 3/20 0.40
CHRM2 P08172 2/20 0.40
CHRM3 P20309 2/20 0.40
ACACB O00763 5/20 0.39
EGFR P00533 1/20 0.37
CHEK2 O96017 1/20 0.37
HRH3 Q9Y5N1 1/20 0.36
P2RX7 Q99572 1/20 0.35
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 2/20 0.35
APP P05067 1/20 0.34
EPHX2 P34913 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6857227 0.90 HRH3 (0.48) AVPR1BACACBHRH3
SCHEMBL6856915 0.90 AVPR1B (0.40) AVPR1B
SCHEMBL6856694 0.89 HRH3 (0.41) AVPR1BACACBHRH3SLC6A4
SCHEMBL6856885 0.88 HRH3 (0.44) AVPR1BACACBHRH3
SCHEMBL6856624 0.88 AVPR1B (0.43) AVPR1BACACBHRH3
SCHEMBL6857457 0.88 HRH1 (0.43) ACACB
SCHEMBL6856447 0.87 ACACB (0.40) AVPR1BACACBHRH3EPHX2
SCHEMBL6857218 0.87 ACACB (0.45) AVPR1BACACBHRH3
SCHEMBL6856195 0.84 MALT1 (0.44) ACACBHRH3EPHX2
SCHEMBL6856761 0.81 AVPR1B (0.41) AVPR1BEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011096461-A1 QUINOLINE DERIVATIVE 大正製薬株式会社 (JP) 2011-08-11 WO disclosed