SCHEMBL6856915

SCHEMBL6856915

COc1cc(-c2nc3ccc(OC4CCNCC4)cc3cc2CC(=O)NC(C)C)ccc1F

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AVPR1B P47901 18/20 0.40
TLR9 Q9NR96 1/20 0.38
TLR8 Q9NR97 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
ACVR1B P36896 1/20 0.37
TGFBR1 P36897 1/20 0.37
ACVR1 Q04771 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6857488 0.90 HRH3 (0.47) AVPR1B
SCHEMBL6856819 0.90 AVPR1B (0.41) AVPR1B
SCHEMBL6856504 0.88 HRH3 (0.43) AVPR1BKCNH2
SCHEMBL6857222 0.87 AVPR1B (0.42) AVPR1BACVR1BTGFBR1ACVR1KCNH2
SCHEMBL6857409 0.82 AVPR1B (0.43) AVPR1B
SCHEMBL6857383 0.81 AVPR1B (0.42) AVPR1B
SCHEMBL6856267 0.79 AVPR1B (0.46) AVPR1B
SCHEMBL6857227 0.79 HRH3 (0.48) AVPR1B
SCHEMBL6857474 0.79 AVPR1B (0.45) AVPR1B
SCHEMBL6856694 0.79 HRH3 (0.41) AVPR1BKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011096461-A1 QUINOLINE DERIVATIVE 大正製薬株式会社 (JP) 2011-08-11 WO disclosed