SCHEMBL6859588

SCHEMBL6859588

CC(NC(=O)C=Cc1cc(F)ccc1F)c1cccc(N2CCOC(CN)C2)c1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNQ2 O43526 2/20 0.51
CYP3A4 P08684 2/20 0.51
KCNQ3 O43525 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP19A1 P11511 1/20 0.51
CYP2C9 P11712 1/20 0.51
ACACB O00763 1/20 0.36
KCNK3 O14649 2/20 0.34
BPTF Q12830 1/20 0.34
NOTUM Q6P988 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6858567 0.89 KCNQ2 (0.56) KCNQ2CYP3A4KCNQ3CYP1A2CYP19A1
SCHEMBL6858570 0.89 KCNQ2 (0.56) KCNQ2CYP3A4KCNQ3CYP1A2CYP19A1
SCHEMBL6858566 0.89 KCNQ2 (0.56) KCNQ2CYP3A4KCNQ3CYP1A2CYP19A1
SCHEMBL6858573 0.89 KCNQ2 (0.56) KCNQ2CYP3A4KCNQ3CYP1A2CYP19A1
SCHEMBL6858584 0.89 KCNQ2 (0.57) KCNQ2CYP3A4KCNQ3CYP1A2CYP19A1
SCHEMBL6858683 0.88 KCNQ2 (0.54) KCNQ2CYP3A4KCNQ3CYP1A2CYP19A1
SCHEMBL6856525 0.83 KCNQ2 (0.54) KCNQ2CYP3A4KCNQ3CYP1A2CYP19A1
SCHEMBL6856512 0.83 KCNQ2 (0.54) KCNQ2CYP3A4KCNQ3CYP1A2CYP19A1
SCHEMBL6856515 0.83 KCNQ2 (0.54) KCNQ2CYP3A4KCNQ3CYP1A2CYP19A1
SCHEMBL6856519 0.83 KCNQ2 (0.54) KCNQ2CYP3A4KCNQ3CYP1A2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6831080-B2 E.g., 3-(2-fluorophenyl)-N-(1-(3-morpholin-4-yl)phenyl)-propyl)acrylamide; disorders responsive to opening of KCNQ potassium channels; analgesics; migraine, bipolar disorders, anticonvulsants, antiepileptic, anxiolytic agents BRISTOL-MYERS SQUIBB COMPANY 2004-12-14 US disclosed