SCHEMBL6859611

SCHEMBL6859611

O=C(c1cccs1)c1nc(N2CCOCC2)nc2ccsc12

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 12/20 0.58
ADORA1 P30542 11/20 0.58
PIK3R1 P27986 1/20 0.57
PIK3CA P42336 1/20 0.57
NPC1 O15118 1/20 0.56
ALDH1A1 P00352 1/20 0.56
TP53 P04637 1/20 0.56
MAPT P10636 1/20 0.56
HPGD P15428 1/20 0.56
RAB9A P51151 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
ALOX5 P09917 3/20 0.48
PTGS2 P35354 3/20 0.48
GAA P10253 1/20 0.47
ADORA2B P29275 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6859506 0.90 ADORA2A (0.62) ADORA2AADORA1PIK3R1PIK3CANPC1
SCHEMBL6859543 0.88 ADORA2A (0.64) ADORA2AADORA1NPC1ALDH1A1RAB9A
SCHEMBL6859739 0.87 ADORA2A (0.59) ADORA2AADORA1PIK3R1PIK3CAADORA2B
SCHEMBL6859687 0.86 ADORA2A (0.58) ADORA2AADORA1PIK3R1PIK3CANPC1
SCHEMBL6852934 0.82 ADORA2A (0.56) ADORA2AADORA1ADORA2B
SCHEMBL6858307 0.82 ADORA2A (0.56) ADORA2AADORA1ADORA2B
SCHEMBL6859714 0.79 ADORA2A (0.53) ADORA2AADORA1ALDH1A1ADORA2B
SCHEMBL6858208 0.79 ADORA2A (0.58) ADORA2AADORA1SMN1; SMN2ADORA2B
SCHEMBL6858206 0.79 ADORA2A (0.58) ADORA2AADORA1SMN1; SMN2ADORA2B
SCHEMBL6852762 0.78 ADORA2A (0.59) ADORA2AADORA1HPGDADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6787541-B1 MOVEMENT DISORDERS, PARKINSON'S DISEASE VERNALIS RESEARCH LIMITED (GB) 2004-09-07 US disclosed