SCHEMBL6859692

SCHEMBL6859692

O=C(c1cccs1)c1nc(N2CCC[C@H]2CO)nc2ccsc12

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 14/20 0.57
ADORA1 P30542 13/20 0.57
ADORA2B P29275 3/20 0.57
ADORA3 P0DMS8 1/20 0.57
ACVR1 Q04771 1/20 0.40
CCNE2 O96020 1/20 0.38
CDK4 P11802 1/20 0.38
CCND1 P24385 1/20 0.38
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38
CD38 P28907 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6852677 1.00 ADORA2A (0.57) ADORA2AADORA1ADORA2BADORA3ACVR1
SCHEMBL6852672 1.00 ADORA2A (0.57) ADORA2AADORA1ADORA2BADORA3ACVR1
SCHEMBL6859554 0.84 ADORA2A (0.54) ADORA2AADORA1ADORA2BADORA3
SCHEMBL6858365 0.83 ADORA2A (0.56) ADORA2AADORA1ADORA2BADORA3ACVR1
SCHEMBL6858361 0.83 ADORA2A (0.56) ADORA2AADORA1ADORA2BADORA3ACVR1
SCHEMBL6859482 0.81 ADORA2A (0.55) ADORA2AADORA1ADORA2BCD38
SCHEMBL6859506 0.80 ADORA2A (0.62) ADORA2AADORA1ADORA2B
SCHEMBL6859687 0.80 ADORA2A (0.58) ADORA2AADORA1ADORA2B
SCHEMBL3678925 0.79 ADORA2A (0.70) ADORA2AADORA1ADORA2BADORA3ACVR1
SCHEMBL3678922 0.79 ADORA2A (0.70) ADORA2AADORA1ADORA2BADORA3ACVR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6787541-B1 MOVEMENT DISORDERS, PARKINSON'S DISEASE VERNALIS RESEARCH LIMITED (GB) 2004-09-07 US disclosed